SCHEMBL3445813

SCHEMBL3445813

CCn1nnc2c(NCc3ccccc3N)nc(NCC(C)N)nc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.50
CCNE1 P24864 9/20 0.50
CDK5 Q00535 4/20 0.48
CCNT1 O60563 3/20 0.48
CDK9 P50750 3/20 0.48
CDK5R1 Q15078 3/20 0.48
CDK7 P50613 2/20 0.48
CCNH P51946 2/20 0.48
CCNE2 O96020 2/20 0.45
CCNA2 P20248 1/20 0.45
CCNA1 P78396 1/20 0.45
AURKA O14965 1/20 0.43
BCDIN3D Q7Z5W3 1/20 0.40
ATM Q13315 1/20 0.39
CDK1 P06493 2/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445380 0.91 CDK2 (0.61) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3446307 0.88 CDK2 (0.49) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3446104 0.87 CDK2 (0.51) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3445762 0.87 CDK2 (0.56) CDK2CCNE1CDK5CDK5R1CCNE2
SCHEMBL3445560 0.85 CCNE1 (0.41) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3445266 0.84 CDK2 (0.40) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3444365 0.83 CDK1 (0.54) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3444369 0.83 CDK1 (0.54) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3446781 0.82 CCNE1 (0.51) CDK2CCNE1CDK5CCNT1CDK9
SCHEMBL3445275 0.82 CDK2 (0.63) CDK2CCNE1CDK5CCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed