SCHEMBL3445946

SCHEMBL3445946

NC(=O)c1cc(C(F)(F)F)ccc1CN1CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.52
MGLL Q99685 2/20 0.50
ABHD6 Q9BV23 1/20 0.50
ALOX5AP P20292 1/20 0.49
FEN1 P39748 1/20 0.49
HIF1A Q16665 5/20 0.48
EPAS1 Q99814 5/20 0.48
CNR2 P34972 3/20 0.47
CNR1 P21554 2/20 0.47
POLB P06746 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.47
FKBP1A P62942 1/20 0.46
FAAH O00519 1/20 0.46
ALDH1A1 P00352 1/20 0.44
THRB P10828 1/20 0.44
IKBKE Q14164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5114802 0.82 SCN9A (0.46) SCN9AMGLLABHD6ALOX5APFEN1
SCHEMBL4996506 0.77 ALDH1A1 (0.63) POLBL3MBTL1HSD17B10ALDH1A1
SCHEMBL2709582 0.77 PDE3B (0.50) SCN9AHIF1AEPAS1CNR2CNR1
SCHEMBL29921818 0.77 PDE3B (0.50) SCN9AHIF1AEPAS1CNR2CNR1
SCHEMBL25026436 0.77 ALOX5AP (0.57) SCN9AMGLLABHD6ALOX5APFEN1
SCHEMBL2228234 0.76 KDM4E (0.58) CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL4506785 0.76 EPHX2 (0.56) ALOX5APFEN1FKBP1A
SCHEMBL27808417 0.76 CYP2C9 (0.51) CNR2CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL24720949 0.76 JAK2 (0.50) HSD17B10ALDH1A1
SCHEMBL11813579 0.75 POLB (0.50) SCN9AHIF1AEPAS1CNR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222165-A1 NOVEL COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS AND USES THEREOF ABBOTT LABORATORIES (US) 2010-09-01 EP claimed
WO-2009067613-A1 NOVEL COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS AND USES THEREOF ABBOTT LABORATORIES (US) 2009-05-28 WO claimed