SCHEMBL3445950

SCHEMBL3445950

COc1cccc(CNc2nc(NCC(C)N)nc3c2nnn3C)c1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.52
CCNE1 P24864 8/20 0.50
CDK2 P24941 8/20 0.50
CCNT1 O60563 3/20 0.50
CDK9 P50750 3/20 0.50
CCNE2 O96020 3/20 0.50
CCNT2 O60583 2/20 0.50
ALDH1A1 P00352 6/20 0.44
MAPT P10636 4/20 0.44
HTT P42858 3/20 0.44
HPGD P15428 2/20 0.44
MEN1 O00255 1/20 0.44
PTBP1 P26599 1/20 0.44
KMT2A Q03164 1/20 0.44
PKM P14618 4/20 0.43
GAA P10253 6/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
ALOX5 P09917 1/20 0.43
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445850 0.92 POLB (0.52) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL3445773 0.92 POLB (0.46) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL3444995 0.90 CCNE1 (0.51) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL3446781 0.89 CCNE1 (0.51) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL15117718 0.85 CDK2 (0.58) CCNE1CDK2CCNT1CDK9CCNE2
SCHEMBL3444312 0.85 CDK2 (0.57) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL3444311 0.85 CDK2 (0.57) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL3444724 0.84 POLB (0.43) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL3446189 0.83 POLB (0.46) POLBCCNE1CDK2CCNT1CDK9
SCHEMBL15117980 0.83 CDK2 (0.72) CCNE1CDK2CCNT1CDK9CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed