SCHEMBL3453534

SCHEMBL3453534

C/C=C\Oc1cncc(N2CCNCC2)c1

nearest known ligand 0.90

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.90
CHRNA4 P43681 9/20 0.90
CHRNA1 P02708 1/20 0.47
CHRNA7 P36544 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3454131 1.00 CHRNB2 (0.90) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL3453535 1.00 CHRNB2 (0.90) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL6347055 0.95 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL5655603 0.95 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL6350045 0.92 CHRNB2 (0.95) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL6358997 0.92 CHRNB2 (0.95) CHRNB2CHRNA4CHRNA1CHRNA7
SCHEMBL5659334 0.85 CHRNB2 (0.76) CHRNB2CHRNA4
SCHEMBL3453243 0.84 CHRNB2 (0.66) CHRNB2CHRNA4
SCHEMBL3453655 0.84 CHRNB2 (0.66) CHRNB2CHRNA4
SCHEMBL3453658 0.84 CHRNB2 (0.66) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1491532-B1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetyloholine receptors NEUROSEARCH AS (DK) 2010-12-15 EP claimed
EP-1491532-B1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetyloholine receptors NEUROSEARCH AS (DK) 2010-12-15 EP disclosed