SCHEMBL3454388

SCHEMBL3454388

COc1cccc(CNC(=O)c2ccc3ccc(C(N)=O)cc3c2)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.70
HPGD P15428 2/20 0.63
LMNA P02545 1/20 0.63
ROCK1 Q13464 3/20 0.60
PRKACA P17612 2/20 0.60
PRKX P51817 2/20 0.60
PRKCQ Q04759 2/20 0.60
ROCK2 O75116 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
GSK3A P49840 1/20 0.60
GSK3B P49841 1/20 0.60
CLK4 Q9HAZ1 1/20 0.60
AURKA O14965 1/20 0.57
ALDH1A1 P00352 2/20 0.57
KDM4E B2RXH2 1/20 0.57
USP2 O75604 1/20 0.57
PLG P00747 1/20 0.56
PLAU P00749 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3038715 0.89 MMP13 (0.72) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL3035661 0.86 MMP13 (0.76) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL3454128 0.86 MMP13 (0.56) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL4499094 0.85 MMP13 (0.74) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL6195092 0.83 MMP13 (0.74) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL5332068 0.83 MMP13 (1.00) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL9416645 0.83 MMP13 (0.94) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL31061610 0.83 MMP13 (1.00) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL31396722 0.81 MMP13 (0.75) MMP13HPGDLMNAROCK1PRKACA
SCHEMBL6658772 0.81 MAPK14 (0.74) MMP13HPGDLMNAROCK1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP disclosed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO disclosed