SCHEMBL3455899

SCHEMBL3455899

Cc1cc2nc(-c3[nH]nc4c3CCN(S(=O)(=O)CC(F)(F)F)C4)[nH]c2cc1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.35
RAB9A P51151 6/20 0.35
ATM Q13315 2/20 0.35
ERAP1 Q9NZ08 1/20 0.35
BRD4 O60885 1/20 0.34
ALDH1A1 P00352 6/20 0.33
MAPT P10636 5/20 0.33
KDM4E B2RXH2 5/20 0.33
SMN1; SMN2 Q16637 5/20 0.33
HPGD P15428 4/20 0.33
KMT2A Q03164 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PPARG P37231 1/20 0.33
NCOA2 Q15596 1/20 0.33
NCOA1 Q15788 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
METAP1 P53582 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3461277 0.90 BRD4 (0.41) NPC1RAB9AATMERAP1BRD4
SCHEMBL3456142 0.87 BRD4 (0.37) NPC1RAB9AATMERAP1BRD4
SCHEMBL3455109 0.85 NPC1 (0.40) NPC1RAB9AATMERAP1BRD4
SCHEMBL3456011 0.85 ALDH1A1 (0.37) NPC1RAB9AATMERAP1BRD4
SCHEMBL3455281 0.84 CNR2 (0.39) NPC1RAB9AATMERAP1BRD4
SCHEMBL3456093 0.84 GUSB (0.38) NPC1RAB9AATMERAP1BRD4
SCHEMBL3458009 0.81 NPC1 (0.39) NPC1RAB9AATMERAP1ALDH1A1
SCHEMBL14031947 0.80 NPC1 (0.40) NPC1RAB9AATMERAP1BRD4
SCHEMBL3458954 0.80 CD4 (0.43) NPC1RAB9AATMERAP1ALDH1A1
SCHEMBL3457131 0.79 GRM5 (0.38) NPC1RAB9AATMERAP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2251340-A1 Substituted tetrahydro-1h-pyrazolo[3,4-c] pyridines, compositions containing same and use thereof Aventis Pharma S.A. (FR) 2010-11-17 EP disclosed
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed