SCHEMBL3456828

SCHEMBL3456828

c1ccc2[nH]c(-c3[nH]nc4c3CCNC4)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.46
ALDH1A1 P00352 9/20 0.46
NPC1 O15118 7/20 0.46
RAB9A P51151 7/20 0.46
HSD17B10 Q99714 5/20 0.46
PKM P14618 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
TP53 P04637 3/20 0.46
ABCB11 O95342 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GAA P10253 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
BTK Q06187 1/20 0.43
FGFR1 P11362 1/20 0.43
FLT1 P17948 1/20 0.43
AURKA O14965 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5067911 0.99 KDM4E (0.45) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL3457670 0.81 ATM (0.40) KDM4ENPC1RAB9AMAPTMETAP2
Hydrochloric Acid SCHEMBL5067947 0.80 ATM (0.39) KDM4ENPC1RAB9ASYKMAPT
SCHEMBL172216 0.67 NPC1 (1.00) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL30634854 0.67 NPC1 (1.00) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL30561047 0.67 NPC1 (1.00) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL7531110 0.66 ALDH1A1 (0.55) KDM4EALDH1A1NPC1RAB9AHSD17B10
Water SCHEMBL9817804 0.65 NPC1 (0.95) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL25425679 0.65 SMN1; SMN2 (0.55) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL29524509 0.65 SMN1; SMN2 (0.55) KDM4EALDH1A1NPC1RAB9AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2251340-A1 Substituted tetrahydro-1h-pyrazolo[3,4-c] pyridines, compositions containing same and use thereof Aventis Pharma S.A. (FR) 2010-11-17 EP disclosed
EP-2251340-A1 Substituted tetrahydro-1h-pyrazolo[3,4-c] pyridines, compositions containing same and use thereof Aventis Pharma S.A. (FR) 2010-11-17 EP disclosed
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed
EP-1646632-A2 SUBSTITUTED TETRAHYDRO-1 I H /I -PYRAZOLO 3,4-C|PYRIDINES, COMPOSITIONS CONTAINING SAME AND USE Aventis Pharma S.A. (FR) 2006-04-19 EP disclosed
WO-2005007653-A2 SUBSTITUTED TETRAHYDRO-1H-PYRAZOLO[3,4-C]PYRIDINES, COMPOSITIONS CONTAINING SAME AND USE AVENTIS PHARMA S.A. (FR) 2005-01-27 WO disclosed