SCHEMBL3457948

SCHEMBL3457948

c1ccc(CNc2nc3ncccc3s2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.50
MAP4K4 O95819 1/20 0.50
PRKCG P05129 1/20 0.50
LYN P07948 1/20 0.50
PRKACA P17612 1/20 0.50
RPS6KB1 P23443 1/20 0.50
AKT1 P31749 1/20 0.50
FLT3 P36888 1/20 0.50
CSNK1D P48730 1/20 0.50
CLK2 P49760 1/20 0.50
IRAK1 P51617 1/20 0.50
PRKX P51817 1/20 0.50
NEK4 P51957 1/20 0.50
PRKCD Q05655 1/20 0.50
ROCK1 Q13464 1/20 0.50
DYRK1A Q13627 1/20 0.50
PKN2 Q16513 1/20 0.50
HIPK4 Q8NE63 1/20 0.50
AURKB Q96GD4 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13540759 0.80 NPC1 (0.60) NPC1RAB9AKMT2AMEN1KDM4E
SCHEMBL1913680 0.78 NPC1 (0.71) ROCK2MAP4K4PRKCGLYNPRKACA
SCHEMBL221983 0.76 SMN1; SMN2 (0.60) NPC1RAB9AKMT2AMEN1LMNA
SCHEMBL14896793 0.74 HRH3 (0.38) NPC1RAB9AKMT2AKDM4ELMNA
SCHEMBL5749417 0.70 NPC1 (0.47) NPC1RAB9AKMT2AMEN1KDM4E
SCHEMBL23965805 0.70 NPC1 (0.60) DYRK1ANPC1RAB9AKMT2AMEN1
SCHEMBL15221710 0.70 CDC7 (0.41) CDC7
SCHEMBL14237602 0.69 FABP1 (0.57) MAP4K4CLK4NPC1RAB9AKMT2A
SCHEMBL5467090 0.69 RORC (0.49) NPC1RAB9AKMT2AMEN1LMNA
SCHEMBL1017978 0.69 KMT2A (0.51) NPC1RAB9AKMT2AMEN1FABP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010435-A2 FUSED OXAZOLE AND THIAZOLE DERIVATIVES AS TRPMS MODULATORS GLENMARK PHARMACEUTICAL S.A. (CH) 2010-01-28 WO disclosed