SCHEMBL3458331

SCHEMBL3458331

Cc1cnc(N)c(-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.52
ADORA1 P30542 1/20 0.52
IKBKB O14920 1/20 0.51
CYP2A6 P11509 2/20 0.49
PIK3CD O00329 1/20 0.48
PIK3CA P42336 1/20 0.48
PIK3CG P48736 1/20 0.48
BRD4 O60885 1/20 0.48
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C19 P33261 1/20 0.45
SCN2A Q99250 2/20 0.44
ATR Q13535 1/20 0.44
PDE10A Q9Y233 1/20 0.44
HRH1 P35367 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
GRIN1 Q05586 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8981695 0.83 MAP4K4 (0.57) CYP2A6PIK3CANPC1RAB9ACYP1A2
SCHEMBL3146889 0.82 ADORA2A (0.52) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL28308461 0.81 ADORA2A (0.54) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL20288103 0.81 CYP2A6 (0.57) ADORA2AADORA1CYP2A6PIK3CDPIK3CA
SCHEMBL2559978 0.79 ADORA2A (0.49) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL10835259 0.79 ADORA2A (0.52) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL9535483 0.78 IKBKB (0.52) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL4412551 0.77 CYP2A6 (0.60) ADORA1CYP2A6NPC1RAB9A
SCHEMBL3140455 0.77 MAP4K4 (0.63) ADORA2AADORA1IKBKBBRD4CYP1A2
SCHEMBL2227047 0.76 MAP4K4 (0.72) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2264010-A1 Hetarylamidines Bayer CropScience AG (DE) 2010-12-22 EP disclosed
EP-2264010-A1 Hetarylamidines Bayer CropScience AG (DE) 2010-12-22 EP disclosed