SCHEMBL28308461

SCHEMBL28308461

Cc1c(-c2cccc(C(F)(F)F)c2)cnc(N)c1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.54
ADORA1 P30542 1/20 0.54
IKBKB O14920 1/20 0.50
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CG P48736 1/20 0.47
BRD4 O60885 1/20 0.47
ATR Q13535 1/20 0.44
SCN2A Q99250 2/20 0.43
KDM1A O60341 1/20 0.43
HRH1 P35367 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C19 P33261 1/20 0.41
IDO1 P14902 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10835259 0.83 ADORA2A (0.52) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL3458331 0.81 ADORA2A (0.52) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL118742 0.78 IKBKB (0.47) ADORA2AADORA1IKBKBBRD4KDM1A
SCHEMBL5327094 0.77 ADORA1 (0.69) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL1388662 0.77 ADORA2A (0.72) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL29655536 0.77 ADORA2A (0.72) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL28736470 0.76 GRIN2B (0.48) ADORA2AADORA1IKBKBPIK3CDPIK3CA
Hydrochloric Acid SCHEMBL27752359 0.75 ADORA2A (0.71) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL3146889 0.75 ADORA2A (0.52) ADORA2AADORA1IKBKBPIK3CDPIK3CA
SCHEMBL15411627 0.75 IKBKB (0.54) ADORA2AADORA1IKBKBPIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114989164-A Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and uses thereof 詹森药业有限公司 2022-09-02 CN disclosed
CN-110062761-B Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and uses thereof 詹森药业有限公司 2022-05-13 CN disclosed
CN-110062761-A Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and their use as GLUN2B receptor modulators 詹森药业有限公司 2019-07-26 CN disclosed