SCHEMBL3463433

SCHEMBL3463433

C=CC(NCc1ccccc1)OC(=O)NC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA7 P43166 1/20 0.42
CA14 Q9ULX7 1/20 0.42
SCN9A Q15858 1/20 0.41
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
RIPK1 Q13546 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
TACR3 P29371 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14763225 0.80 SCN9A (0.47) ALDH1A1CYP3A4CYP2C9CYP2C19SCN9A
SCHEMBL14763226 0.80 SCN9A (0.47) ALDH1A1CYP3A4CYP2C9CYP2C19SCN9A
SCHEMBL3463367 0.79 SMN1; SMN2 (0.43) CYP2C9CYP2C19MAPTSMN1; SMN2
SCHEMBL28450250 0.74 ATM (0.51) ALDH1A1CA12CA1CA7CA14
SCHEMBL29253631 0.74 KMT2A (0.56) CA12CA1CA7CA14SCN9A
SCHEMBL29253670 0.74 KMT2A (0.56) CA12CA1CA7CA14SCN9A
SCHEMBL27496212 0.72 SCN9A (0.47) SCN9ARAB9ANPC1MAPTATM
SCHEMBL395106 0.72 SCN9A (0.47) SCN9ARAB9ANPC1MAPTATM
SCHEMBL395107 0.72 SCN9A (0.47) SCN9ARAB9ANPC1MAPTATM
SCHEMBL28359858 0.70 SCN9A (0.48) CYP3A4CA12CA1CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010435-A2 FUSED OXAZOLE AND THIAZOLE DERIVATIVES AS TRPMS MODULATORS GLENMARK PHARMACEUTICAL S.A. (CH) 2010-01-28 WO disclosed