SCHEMBL3467482

SCHEMBL3467482

CCOc1ccc2nc(NC(=O)c3cn(CCCCCC(=O)NO)c4ccccc4c3=O)sc2c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.52
SMN1; SMN2 Q16637 8/20 0.52
TP53 P04637 3/20 0.52
RAB9A P51151 10/20 0.51
NPC1 O15118 9/20 0.51
HSD17B10 Q99714 2/20 0.51
KMT2A Q03164 4/20 0.51
PKM P14618 2/20 0.51
NPSR1 Q6W5P4 2/20 0.51
OPRK1 P41145 1/20 0.51
MEN1 O00255 3/20 0.49
PSMD14 O00487 1/20 0.49
USP2 O75604 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HTT P42858 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HSP90AA1 P07900 1/20 0.49
HPGD P15428 1/20 0.49
ALOX15 P16050 1/20 0.49
CSNK1D P48730 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467494 0.87 HDAC1 (0.55) MAPTKMT2AMEN1HDAC1HDAC6
SCHEMBL3468955 0.84 NPC1 (0.51) MAPTSMN1; SMN2RAB9ANPC1KMT2A
SCHEMBL3467572 0.80 HDAC1 (0.51) MAPTTP53KMT2AMEN1HDAC1
SCHEMBL3467367 0.80 CNR2 (0.51) MAPTKMT2AMEN1HTTHDAC1
SCHEMBL3467882 0.79 HDAC1 (0.50) MAPTRAB9ANPC1HTTKDM4E
SCHEMBL7926022 0.77 HPGD (0.53) SMN1; SMN2HSD17B10NPSR1ALDH1A1HPGD
SCHEMBL3467299 0.76 HDAC1 (0.53) MAPTKMT2AMEN1HDAC1HDAC6
SCHEMBL3468762 0.76 HDAC1 (0.51) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL3468139 0.76 CNR2 (0.58) KMT2AMEN1HDAC1HDAC6HDAC3
SCHEMBL3467928 0.74 HDAC1 (0.60) HDAC1HDAC6HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010073078-A2 HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LTD. (IN) 2010-07-01 WO disclosed