SCHEMBL3473180

SCHEMBL3473180

c1ccc(C[C@@H]2CCCNC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EED O75530 4/20 0.61
GBA1 P04062 1/20 0.61
KMT2A Q03164 1/20 0.53
HRH4 Q9H3N8 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
CHRNB2 P17787 3/20 0.48
CHRNA4 P43681 3/20 0.48
POLB P06746 1/20 0.47
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547993 1.00 EED (0.61) EEDGBA1KMT2AHRH4HRH3
SCHEMBL1761058 1.00 EED (0.61) EEDGBA1KMT2AHRH4HRH3
Hydrochloric Acid SCHEMBL3914926 0.98 EED (0.60) EEDGBA1KMT2AHRH4HRH3
Hydrochloric Acid SCHEMBL7068731 0.96 EED (0.58) EEDGBA1KMT2AHRH4HRH3
SCHEMBL9598369 0.95 GBA1 (0.59) EEDGBA1KMT2AHRH4HRH3
Cyclooctanamine SCHEMBL4971880 0.89 EED (0.52) EEDGBA1KMT2AHRH4HRH3
SCHEMBL4892499 0.89 GBA1 (0.78) EEDGBA1HRH4HRH3POLB
SCHEMBL892689 0.89 GBA1 (0.78) EEDGBA1HRH4HRH3POLB
SCHEMBL4889591 0.89 GBA1 (0.78) EEDGBA1HRH4HRH3POLB
SCHEMBL13576621 0.86 EED (0.59) EEDGBA1KMT2AHRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069979-A1 PYRAN DERIVATIVES AS CCR3 MODULATORS NYCOMED GMBH (DE) 2010-06-24 WO disclosed
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed