SCHEMBL3473755

SCHEMBL3473755

COc1ccc(C/C=N/N(C)c2cc(=O)n(C)c(=O)[nH]2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.55
KDM4C Q9H3R0 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 5/20 0.49
HPGD P15428 3/20 0.49
THRB P10828 2/20 0.49
PKM P14618 3/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.41
NR1I2 O75469 1/20 0.41
AHR P35869 1/20 0.41
DAO P14920 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 3/20 0.39
CASP1 P29466 1/20 0.37
BRCA1 P38398 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
G6PD P11413 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179271 0.82 KDM4E (0.75) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2179274 0.82 KDM4E (0.75) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL3470482 0.74 ALDH1A1 (0.63) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2182131 0.73 SMN1; SMN2 (0.61) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2182128 0.73 SMN1; SMN2 (0.61) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2182121 0.70 KDM4E (0.61) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2182123 0.70 KDM4E (0.61) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2182930 0.70 ALDH1A1 (0.59) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL2182936 0.70 ALDH1A1 (0.59) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD
SCHEMBL3474190 0.70 SMN1; SMN2 (0.55) KDM4EKDM4CSMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed