SCHEMBL3475461

SCHEMBL3475461

NC(=O)N(c1ccccc1)c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.47
HTT P42858 3/20 0.47
PTGIR P43119 1/20 0.46
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 4/20 0.42
POLB P06746 3/20 0.42
KMT2A Q03164 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
RECQL P46063 1/20 0.42
BLM P54132 1/20 0.42
MCL1 Q07820 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
LMNA P02545 1/20 0.41
NAPRT Q6XQN6 1/20 0.41
P4HTM Q9NXG6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726837 0.89 HTT (0.53) NPSR1HTTTP53TSHRALDH1A1
SCHEMBL28021427 0.87 HTT (0.43) NPSR1HTTTP53TSHRALDH1A1
SCHEMBL28021882 0.87 ALDH1A1 (0.45) NPSR1HTTPTGIRTP53ALDH1A1
SCHEMBL28021440 0.87 HTT (0.43) NPSR1HTTPTGIRTP53TSHR
SCHEMBL10855054 0.85 NPSR1 (0.50) NPSR1HTTPTGIRTP53TSHR
SCHEMBL5271141 0.85 MEN1 (0.45) NPSR1HTTPTGIRTSHRALDH1A1
SCHEMBL10668533 0.84 NPSR1 (0.63) NPSR1HTTPTGIRTP53TSHR
SCHEMBL9742065 0.83 NPSR1 (0.50) NPSR1HTTTSHRALDH1A1POLB
SCHEMBL27511353 0.83 NPC1 (0.42) NPSR1HTTPTGIRTP53ALDH1A1
SCHEMBL27551941 0.83 HTT (0.47) NPSR1HTTPTGIRTP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4173701-A None JP disclosed
JP-58194804-A None JP disclosed
CN-111072559-B Construction and application of 2, 6-dibromopyridine oxidation system 浙江工商大学 2021-06-18 CN disclosed
CN-111072559-A Construction and application of 2, 6-dibromopyridine oxidation system 浙江工商大学 2020-04-28 CN disclosed
CN-103880738-A Preparation method of 1-(2-chloro-4-pyridyl)-3-phenylurea ZHEJIANG TIDE CROP TECHNOLOGY CO LTD 2014-06-25 CN disclosed
CN-103880737-A Preparation method of 1-(2-chloro-4-pyridyl)-3-phenylurea ZHEJIANG TIDE CROP TECHNOLOGY CO LTD 2014-06-25 CN disclosed
WO-2010131030-A1 PYRIDYLUREA DERIVATIVES AND THEIR THERAPEUTIC USE PULMAGEN THERAPEUTICS (INFLAMMATION) LIMITED (GB) 2010-11-18 WO disclosed
CN-1626517-A Method of synthesized pyridyl of substituting ramification in urea class DALIAN CHEMICAL PHYSICS INST (CN) 2005-06-15 CN disclosed
CN-1181058-C Process for preparing pyridylphenylureas 四川省兰月科技开发公司 2004-12-22 CN disclosed
CN-1156450-C Process for preparing unsymmetric phenylpyridyl substances 中国科学院大连化学物理研究所 2004-07-07 CN disclosed
CN-1368500-A Process for preparing unsymmetric phenylpyridyl substances DALIAN CHEMICAL PHYSICS INST (CN) 2002-09-11 CN disclosed
US-6242257-B1 CUTTING APICAL EXPLANT FROM GERMINATED COTTON SEEDLING, CULTURING FOR SHOOT PROLIFERATION IN MEDIUM FREE OF AUXIN AND SUCROSE, HARVESTING SHOOTS, THEN CULTURING EACH SHOOT IN SECOND MEDIUM; EFFICIENT PROCESS FOR GENETIC ENGINEERING COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2001-06-05 US disclosed
US-6133299-A ADMINISTERING TO A MAMMAL A COMPOUND SELECTED FROM RALITOLINE, PHENYTOIN, LAMOTRIGINE, CARBAMAZEPINE, LIDOCAINE OR TETRODOTOXIN; TREATING DISEASE SUCH AS STROKE, ALZHEIMER'S DISEASE, HUNTINGTON'S DISEASE, PARKINSON'S DISEASE WARNER-LAMBERT COMPANY (US) 2000-10-17 US disclosed
US-5569765-A 2-anilinopyridine pesticides BASF AKTIENGESELLSCHAFT (DE) 1996-10-29 US disclosed
US-5453432-A Anilinopyridines BASF AKTIENGESELLSCHAFT (DE) 1995-09-26 US disclosed
WO-1994018972-A2 METHODS FOR TREATING NEURODEGENERATIVE DISEASES AND DISORDERS USING N-(2,6-DISUBSTITUTED AROMATIC)-N'-PYRIDINYL UREAS AND OTHER ANTICONVULSANT COMPOUNDS WARNER-LAMBERT COMPANY (US) 1994-09-01 WO disclosed
US-5154751-A HERBICIDAL UREA COMPOUNDS AND COMPOSITIONS CIBA-GEIGY CORPORATION (US) 1992-10-13 US disclosed
JP-H04173701-A CHEMICAL INJURY-MITIGATIVE AGENT FOR PADDY HERBICIDE HOKKO CHEM IND CO LTD 1992-06-22 JP disclosed
EP-0233040-A2 Stigma of crocus sativus L. and method for the production thereof AJINOMOTO CO., INC. (JP) 1987-08-19 EP disclosed
JP-S58194804-A AGENT FOR INCREASING YIELD OF POTATO AND TARO OKAMOTO TOSHIHIKO 1983-11-12 JP disclosed