Sulconazole

Sulconazole

SCHEMBL34761

Clc1ccc(CSC(Cn2ccnc2)c2ccc(Cl)cc2Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Sulconazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 10/20 1.00
CYP3A4 P08684 9/20 1.00
CYP2C9 P11712 9/20 1.00
CYP1A2 P05177 6/20 1.00
CYP2D6 P10635 6/20 1.00
CYP2C19 P33261 6/20 1.00
TDP1 Q9NUW8 4/20 1.00
NR1I2 O75469 4/20 1.00
ADORA3 P0DMS8 4/20 1.00
ADRA2B P18089 4/20 1.00
CHRM3 P20309 4/20 1.00
SLC6A2 P23975 4/20 1.00
SLC6A4 P31645 4/20 1.00
DRD3 P35462 4/20 1.00
OPRK1 P41145 4/20 1.00
KCNH2 Q12809 4/20 1.00
USP2 O75604 3/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
ADRA2C P18825 3/20 1.00
ALOX15 P16050 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulconazole SCHEMBL34762 1.00 IDO1 (1.00) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
Sulconazole SCHEMBL22123404 1.00 IDO1 (1.00) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
Sulconazole SCHEMBL29923838 1.00 IDO1 (1.00) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
Sulconazole SCHEMBL7600689 1.00 IDO1 (1.00) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
Sulconazole SCHEMBL7600685 1.00 IDO1 (1.00) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
Sulconazole SCHEMBL29194304 0.99 IDO1 (0.98) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
Sulconazole SCHEMBL28462757 0.99 IDO1 (0.98) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL11698496 0.93 IDO1 (0.87) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL11699369 0.93 IDO1 (0.87) IDO1CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL11693931 0.93 IDO1 (0.87) IDO1CYP3A4CYP2C9CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 13412 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122005693-A Application of Jiaweidanzhi Xiaoyao powder or extract thereof in preparation of medicines for treating depression complicated with ulcerative colitis 河南中医药大学 2026-05-12 CN claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260102419-A1 USE OF COMPOUNDS IN THE TREATMENT OF FUNGAL INFECTIONS BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL (CH) 2026-04-16 US claimed
EP-4719384-A2 COMPOUNDS WITH ANTIFUNGAL PROPERTIES Trustees of Dartmouth College (US) 2026-04-08 EP claimed
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
EP-4676500-A2 MICROBIAL CONSORTIA Kanvas Biosciences, Inc (US) 2026-01-14 EP claimed
US-20260007753-A1 DERMAL SKIN PROTECTANT AND CARRIER INSPIRED MAT STRATEGIES LLC (US) 2026-01-08 US claimed
US-20250387371-A1 COMPOSITIONS AND FORMULATION METHODS FOR SUSTAINED LOCAL RELEASE OF ANTIFIBROTICS THE HOPKINS UNIVERISTY (US) 2025-12-25 US claimed
EP-4659014-A1 EMULSION-BASED THICK-FILM ANTIFOULING COATING FOR HIGHLY SENSITIVE ELECTROCHEMICAL SENSING President And Fellows Of Harvard College (US) 2025-12-10 EP claimed
US-12419959-B2 Dermal skin protectant and carrier Inspired Material Strategies, LLC (US) 2025-09-23 US claimed
EP-0310122-B1 ANTIFUNGAL COMPOSITION KAKEN PHARMACEUTICAL CO., LTD. (JP) 1991-07-24 EP claimed
US-5028418-A Miconazole, Econazole, Sulconazole BRISTOL-MYERS SQUIBB COMPANY (US) 1991-07-02 US claimed
US-5002938-A Fungicide, Steroid, Alcohol and Diol and/or Triol Solvent, Hydroxyalkyl Cellulose BRISTOL-MYERS SQUIBB COMPANY (US) 1991-03-26 US claimed
WO-1991002497-A1 TOPICAL NIFEDIPINE FOR CUTANEOUS, OCULAR, MUCOSAL HYPERSENSITIVITY, INFLAMMATORY AND HYPERPROLIFERATIVE CONDITIONS BETH ISRAEL HOSPITAL ASSOCIATION (US) 1991-03-07 WO claimed
WO-1991002527-A1 METHOD AND COMPOSITION FOR THE TREATMENT OF CUTANEOUS, OCULAR, AND MUCOSAL HYPERSENSITIVITY, INFLAMMATION, AND HYPERPROLIFERATIVE CONDITIONS USING TOPICAL PREPARATIONS OF SEROTONIN ANTAGONISTS BETH ISRAEL HOSPITAL ASSOCIATION (US) 1991-03-07 WO claimed
EP-0310122-A1 Antifungal composition KAKEN PHARMACEUTICAL CO., LTD. (JP) 1989-04-05 EP claimed
EP-0064283-B1 STABILIZATION OF 1-SUBSTITUTED IMIDAZOLE DERIVATIVES IN TALC SYNTEX (U.S.A.) INC. (US) 1987-01-28 EP claimed
US-4277475-A FOR BOTH MALES AND FEMALES SYNTEX (U.S.A.) INC. (US) 1981-07-07 US claimed
US-4247552-A Contraceptive compositions and methods employing 1-substituted imidazole derivatives SYNTEX (U.S.A.) INC. (US) 1981-01-27 US claimed
US-4055652-A 1-[β(R-thio)phenethyl]imidazoles and derivatives thereof SYNTEX (U.S.A.) INC. (US) 1977-10-25 US claimed