SCHEMBL3477262

SCHEMBL3477262

CNC(=O)c1cccc(Cl)c1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.53
TSHR P16473 1/20 0.48
DOT1L Q8TEK3 1/20 0.48
PLK1 P53350 1/20 0.47
ALDH1A1 P00352 3/20 0.47
GAA P10253 1/20 0.46
POLB P06746 1/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
USP2 O75604 1/20 0.44
MT-CO2 P00403 1/20 0.44
LMNA P02545 1/20 0.44
TTR P02766 1/20 0.44
PLA2G1B P04054 1/20 0.44
CYP1A2 P05177 1/20 0.44
PGR P06401 1/20 0.44
CYP3A4 P08684 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
ADORA3 P0DMS8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3780962 0.89 DOT1L (0.50) PBRM1TSHRDOT1LPLK1ALDH1A1
SCHEMBL27497363 0.84 DOT1L (0.47) PBRM1TSHRDOT1LPLK1ALDH1A1
SCHEMBL29040264 0.84 PBRM1 (0.54) PBRM1TSHRALDH1A1GAAPOLB
SCHEMBL25364346 0.82 PBRM1 (0.53) PBRM1TSHRALDH1A1POLBKMT2A
SCHEMBL551796 0.81 PBRM1 (0.49) PBRM1TSHRALDH1A1POLBKMT2A
SCHEMBL31356504 0.81 TSHR (0.65) PBRM1TSHRALDH1A1POLBKMT2A
SCHEMBL275485 0.81 TSHR (0.65) PBRM1TSHRALDH1A1POLBKMT2A
SCHEMBL4157657 0.81 DOT1L (0.56) DOT1LALDH1A1GAAPOLBKMT2A
SCHEMBL4143751 0.79 TAS1R3 (0.60) TSHRPLK1ALDH1A1GAAPOLB
SCHEMBL6640962 0.79 TSHR (0.53) PBRM1TSHRALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113754621-B Synthesis method of 2,3',3,4' -diphenyl sulfone tetracarboxylic dianhydride 常州市阳光药业有限公司 2023-06-23 CN claimed
EP-2233512-B1 POLYTHIOETHERIMIDES AND METHOD FOR PRODUCING THEREOF NINGBO INST MATERIALS TECHNOLOGY & ENG CAS (CN) 2013-03-20 EP claimed
US-20110065891-A1 POLYTHIOETHERIMIDES AND METHOD FOR PRODUCING THEREOF CHANGCHUN HIPOLYKING CO.,LTD. (CN) 2011-03-17 US claimed
EP-2233512-A1 POLYTHIOETHERIMIDES AND METHOD FOR PRODUCING THEREOF Ningbo Institute Of Materials Technology And Engineering, Chinese Academy Of Sciences (CN) 2010-09-29 EP claimed
CN-113754621-B Synthesis method of 2,3',3,4' -diphenyl sulfone tetracarboxylic dianhydride 常州市阳光药业有限公司 2023-06-23 CN disclosed
EP-2233512-B1 POLYTHIOETHERIMIDES AND METHOD FOR PRODUCING THEREOF NINGBO INST MATERIALS TECHNOLOGY & ENG CAS (CN) 2013-03-20 EP disclosed
US-20110065891-A1 POLYTHIOETHERIMIDES AND METHOD FOR PRODUCING THEREOF CHANGCHUN HIPOLYKING CO.,LTD. (CN) 2011-03-17 US disclosed
EP-2233512-A1 POLYTHIOETHERIMIDES AND METHOD FOR PRODUCING THEREOF Ningbo Institute Of Materials Technology And Engineering, Chinese Academy Of Sciences (CN) 2010-09-29 EP disclosed
CN-100519545-C 2,3',3,4'-diphenyl sulfide tetracarboxylic dianhydride CHANGCHUN APPLIED CHEMISTRY (CN) 2009-07-29 CN disclosed
CN-1724528-A 2,3 ', 3,4 '-preparation method of diphenyl sulfide tetracarboxylic dianhydride CHANGCHUN INST OF APPLIED CHEN (CN) 2006-01-25 CN disclosed