SCHEMBL3483033

SCHEMBL3483033

CC(O)CNC(=O)c1ccc(-c2ccn3ncc(/C=C4\NC(=O)NC4=O)c3n2)s1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PRF1 P14222 2/20 0.42
CAMK2D Q13557 10/20 0.34
KCNH2 Q12809 2/20 0.34
CSNK2B P67870 2/20 0.34
NTRK1 P04629 5/20 0.32
JAK2 O60674 4/20 0.32
AKT3 Q9Y243 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12979332 1.00 PRF1 (0.42) PRF1CAMK2DKCNH2CSNK2BNTRK1
SCHEMBL3483036 1.00 PRF1 (0.42) PRF1CAMK2DKCNH2CSNK2BNTRK1
SCHEMBL12979612 0.85 DYRK1A (0.35) CAMK2DCSNK2BNTRK1JAK2
SCHEMBL860754 0.85 DYRK1A (0.35) CAMK2DCSNK2BNTRK1JAK2
SCHEMBL860753 0.85 DYRK1A (0.35) CAMK2DCSNK2BNTRK1JAK2
SCHEMBL12979532 0.85 SMN1; SMN2 (0.34) CAMK2DKCNH2CSNK2BAKT3
SCHEMBL12979694 0.85 SMN1; SMN2 (0.34) CAMK2DKCNH2CSNK2BAKT3
SCHEMBL12979020 0.84 CAMK2D (0.39) CAMK2DKCNH2NTRK1JAK2AKT3
SCHEMBL14679098 0.82 CAMK2D (0.34) PRF1CAMK2DKCNH2NTRK1JAK2
SCHEMBL12584199 0.82 CSNK2B (0.39) PRF1CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367681-B2 Pyrazolopyrimidines and related heterocycles as kinase inhibitors CYLENE PHARMACEUTICALS, INC. (US) 2013-02-05 US disclosed
US-8367681-B2 Pyrazolopyrimidines and related heterocycles as kinase inhibitors CYLENE PHARMACEUTICALS, INC. (US) 2013-02-05 US disclosed
US-8367681-B2 Pyrazolopyrimidines and related heterocycles as kinase inhibitors CYLENE PHARMACEUTICALS, INC. (US) 2013-02-05 US disclosed
US-20100331314-A1 PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS SENHWA BIOSCIENCES, INC. (TW) 2010-12-30 US disclosed
US-20100331314-A1 PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS SENHWA BIOSCIENCES, INC. (TW) 2010-12-30 US disclosed
US-20100331314-A1 PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS SENHWA BIOSCIENCES, INC. (TW) 2010-12-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331314-A1 PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS PIM1, PIM2, PIM3 PRF1 2051/4885CAMK2D 258/4885KCNH2 959/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.