SCHEMBL3495835

SCHEMBL3495835

CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCCO[C@@H](CO)COC(=O)CCCCCCCCCCCCCCCCC

nearest known ligand 0.80

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.80
CNR2 P34972 3/20 0.80
PRKCA P17252 3/20 0.71
PRKCE Q02156 2/20 0.71
PRKCQ Q04759 2/20 0.71
PRKCD Q05655 2/20 0.71
ALDH1A1 P00352 2/20 0.67
FAAH O00519 3/20 0.64
DGKA P23743 1/20 0.63
MAPT P10636 1/20 0.61
HPGD P15428 1/20 0.61
MGLL Q99685 1/20 0.59
SELP P16109 1/20 0.59
S1PR1 P21453 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5407956 1.00 CNR1 (0.80) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL7192929 1.00 CNR1 (0.80) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL7192934 1.00 CNR1 (0.80) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL10492090 1.00 CNR1 (0.80) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL10492106 0.96 CNR1 (0.75) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL10492119 0.96 PRKCA (0.76) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL1145290 0.96 PRKCA (0.76) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL7557200 0.96 PRKCA (0.76) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL7557194 0.96 PRKCA (0.76) CNR1CNR2PRKCAPRKCEPRKCQ
SCHEMBL29644755 0.96 PRKCA (0.76) CNR1CNR2PRKCAPRKCEPRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100152277-A1 DIACYLGLYCEROL ACYLTRANSFERASE ASSAY JANSSEN PHARMACEUTICA N.V. (BE) 2010-06-17 US claimed
EP-1831393-A1 DIACYLGLYCEROL ACYLTRANSFERASE ASSAY JANSSEN PHARMACEUTICA N.V. (BE) 2007-09-12 EP claimed
WO-2006067071-A1 DIACYLGLYCEROL ACYLTRANSFERASE ASSAY JANSSEN PHARMACEUTICA N.V. (BE) 2006-06-29 WO claimed
US-20030171277-A1 Orally administered peptides to ameliorate atherosclerosis THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-09-11 US claimed
CN-121007977-A Biomarker combination for liver cancer diagnosis and application thereof 香港中文大学 2025-11-25 CN disclosed
US-20100152277-A1 DIACYLGLYCEROL ACYLTRANSFERASE ASSAY JANSSEN PHARMACEUTICA N.V. (BE) 2010-06-17 US disclosed
US-6566047-B1 Detecting modulator of neuron propagation; obtain neurons, incubate with modulator, monitor adjustment in neuron activity, evaluate neuron migration THE REGENTS OF THE UNIVERSITY OF COLORADO 2003-05-20 US disclosed
US-6221658-B1 NUCLEOTIDE SEQUENCE; FOR DECREASING INTRACELLULAR LEVELS OF DIACYLGLYCEROL AND INCREASING INTRACELLULAR LEVELS OF PHOSPHATIDIC ACID IN A EUKARYOTIC CELL UNIVERSITY OF UTAH RESEARCH FOUNDATION 2001-04-24 US disclosed
WO-1999061585-A1 ASSAYS FOR IDENTIFYING ANTI-METASTATIC AND NEURITE-PROMOTING AGENTS AND USES THEREOF UNIVERSITY TECHNOLOGY CORPORATION (US) 1999-12-02 WO disclosed
US-5976875-A NUCLEIC ACID WHICH CODES FOR ENZYME IMPORTANT IN CELL MEMBRANE AND TRIGLYCERIDE FORMATION AND PROTEIN KINASE C ACTIVATION; DECREASING INTRACELLULAR LEVELS OF DIACYLGLYCEROL AND INCREASING INTRACELLULAR LEVELS OF PHOSPHATIDIC ACID UNIVERSITY OF UTAH (US) 1999-11-02 US disclosed
US-5512429-A Assay for enzyme activity BRITISH TECHNOLOGY GROUP LIMITED (GB) 1996-04-30 US disclosed
EP-0493426-B1 ASSAY FOR ENZYME ACTIVITY BRITISH TECH GROUP (GB) 1995-11-08 EP disclosed
WO-1991004338-A1 ASSAY FOR ENZYME ACTIVITY BRITISH TECHNOLOGY GROUP PLC (GB) 1991-04-04 WO disclosed