SCHEMBL3497477

SCHEMBL3497477

N#C[C@H](O)c1ccccc1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
TRPA1 O75762 1/20 0.35
DYRK1A Q13627 1/20 0.35
HTT P42858 1/20 0.35
CXCR2 P25025 3/20 0.34
CFTR P13569 2/20 0.34
CXCR1 P25024 2/20 0.34
OPRL1 P41146 2/20 0.33
CCR1 P32246 1/20 0.33
SLC18A3 Q16572 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
ADRB3 P13945 1/20 0.31
TSPO P30536 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL198230 1.00 TSHR (0.50) TSHRIDO1TDO2TRPA1DYRK1A
SCHEMBL6687100 1.00 TSHR (0.50) TSHRIDO1TDO2TRPA1DYRK1A
SCHEMBL13937393 0.84 TSHR (0.61) TSHRTRPA1ALDH1A1L3MBTL1
SCHEMBL7351692 0.78 TSHR (0.50) TSHRHTTCCR1ALDH1A1CYP3A4
SCHEMBL29413826 0.78 CFTR (0.37) TSHRIDO1TDO2HTTCFTR
SCHEMBL3372946 0.76 IDO1 (0.43) TSHRIDO1TDO2HTTCFTR
SCHEMBL11604556 0.76 IDO1 (0.43) TSHRIDO1TDO2HTTCFTR
SCHEMBL5117680 0.76 IDO1 (0.43) TSHRIDO1TDO2HTTCFTR
SCHEMBL5117761 0.76 IDO1 (0.43) TSHRIDO1TDO2HTTCFTR
SCHEMBL3375814 0.76 IDO1 (0.43) TSHRIDO1TDO2HTTCFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105296512-A Nitrilases, nucleic acids encoding them and methods for making and using them BASF ENZYMES LLC 2016-02-03 CN disclosed
EP-2465929-B1 R-HNL random variants and their use for preparing optically pure, sterically hindered cyanohydrins DSM IP ASSETS BV (NL) 2015-12-02 EP disclosed
CN-102796750-B The nucleic acid of nitrilase, encoding nitrilase enzyme, and the method preparing and use them BASF ENZYMES LLC (US) 2015-09-16 CN disclosed
US-8846366-B2 R-hydroxynitrile lyase (R-HNL) random variants and their use for preparing optically pure, sterically hindered cyanohydrins DSM IP ASSETS BV (NL) 2014-09-30 US disclosed
CN-1849391-B Nitrilases, nucleic acids encoding nitrilases, and methods of making and using the same DIVERSA CORP 2014-06-11 CN disclosed
EP-2092060-B1 R-HNL RANDOM VARIANTS AND THEIR USE FOR PREPARING OPTICALLY PURE, STERICALLY HINDERED CYANOHYDRINS DSM IP ASSETS BV (NL) 2014-01-22 EP disclosed
EP-2465929-A1 R-HNL random variants and their use for preparing optically pure, sterically hindered cyanohydrins DSM IP Assets B.V. (NL) 2012-06-20 EP disclosed
US-20100143986-A1 R-HNL RANDOM VARIANTS AND THEIR USE FOR PREPARING OPTICALLY PURE, STERICALLY HINDERED CYANOHYDRINS DSM IP ASSETS BV (NL) 2010-06-10 US disclosed
EP-2092060-A1 R-HNL RANDOM VARIANTS AND THEIR USE FOR PREPARING OPTICALLY PURE, STERICALLY HINDERED CYANOHYDRINS DSMIP Assets B.V. (NL) 2009-08-26 EP disclosed
WO-2008071695-A1 R-HNL RANDOM VARIANTS AND THEIR USE FOR PREPARING OPTICALLY PURE, STERICALLY HINDERED CYANOHYDRINS DSM IP ASSETS BV (NL) 2008-06-19 WO disclosed
CN-1849391-A Nitrilases, nucleic acids encoding nitrilases, and methods of making and using the same DIVERSA CORP (US) 2006-10-18 CN disclosed