SCHEMBL3510402

SCHEMBL3510402

CC(C)(C)OC(=O)Nc1cccc(-c2ccc(C(=O)O)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.67
RXRA P19793 2/20 0.54
RXRB P28702 2/20 0.54
HDAC1 Q13547 3/20 0.51
HDAC4 P56524 2/20 0.51
ADORA3 P0DMS8 1/20 0.50
HDAC3 O15379 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
BCL2 P10415 1/20 0.49
BECN1 Q14457 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13754832 0.90 CYP17A1 (0.64) CYP17A1HDAC1HDAC4ADORA3HDAC3
SCHEMBL25432469 0.86 CYP17A1 (0.55) CYP17A1RXRARXRBMEN1NPC1
SCHEMBL3360413 0.86 CYP17A1 (0.63) CYP17A1RXRARXRBBCL2BECN1
SCHEMBL3789848 0.85 CYP17A1 (0.62) CYP17A1HDAC1HDAC4HDAC3HDAC2
SCHEMBL29435026 0.84 HDAC3 (0.58) CYP17A1HDAC1HDAC3HDAC2HDAC8
SCHEMBL222876 0.84 HDAC3 (0.58) CYP17A1HDAC1HDAC3HDAC2HDAC8
SCHEMBL7439456 0.83 HDAC3 (0.57) CYP17A1HDAC1HDAC3HDAC2HDAC8
SCHEMBL12740173 0.83 CYP17A1 (0.60) CYP17A1HDAC1HDAC4HDAC3HDAC2
SCHEMBL1684366 0.83 CYP17A1 (0.60) CYP17A1HDAC1HDAC4HDAC3HDAC2
SCHEMBL31671045 0.82 CYP17A1 (0.76) CYP17A1HDAC1HDAC4HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286035-A1 NEUROMEDIN U DERIVATIVE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286035-A1 NEUROMEDIN U DERIVATIVE NMUR1, NMUR2, NMBR CYP17A1 4511/4885RXRA 4340/4885RXRB 4240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.