SCHEMBL3515574

SCHEMBL3515574

COc1ccc(-c2ccnc(Nc3ccc(S(=O)(=O)NCCN(C)C)cc3)n2)cc1F

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 7/20 0.64
CDK2 P24941 6/20 0.57
CDK4 P11802 3/20 0.54
CDK1 P06493 1/20 0.54
CCNT1 O60563 7/20 0.48
CDK9 P50750 7/20 0.48
CCNA2 P20248 1/20 0.47
CDK6 Q00534 1/20 0.47
CHUK O15111 1/20 0.46
NEK1 Q96PY6 1/20 0.46
PLK1 P53350 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3521750 0.95 IKBKB (0.65) IKBKBCDK2CDK4CDK1CCNT1
Acetic Acid SCHEMBL4877880 0.91 IKBKB (0.60) IKBKBCDK2CDK4CDK1CCNT1
SCHEMBL3519883 0.91 IKBKB (0.52) IKBKBCDK2CDK4CDK1CDK9
SCHEMBL3522199 0.90 IKBKB (0.65) IKBKBCDK2CDK4CDK1CCNT1
SCHEMBL3516749 0.90 IKBKB (0.51) IKBKBCDK2CDK4CDK1CCNT1
SCHEMBL3516415 0.88 IKBKB (0.59) IKBKBCDK2CDK4CDK1CCNT1
SCHEMBL3516533 0.88 IKBKB (0.66) IKBKBCDK2CDK4CDK1CCNA2
SCHEMBL3516904 0.88 IKBKB (0.49) IKBKBCDK2CDK4CDK1CCNT1
SCHEMBL3521141 0.88 IKBKB (0.49) IKBKBCDK2CDK4CDK1
SCHEMBL3521916 0.86 IKBKB (0.47) IKBKBCDK2CDK4CDK1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799915-B2 Anilino-pyrimidine analogs WYETH LLC (US) 2010-09-21 US claimed
US-20060079543-A1 Anilino-pyrimidine analogs WYETH (US) 2006-04-13 US claimed
US-7799915-B2 Anilino-pyrimidine analogs WYETH LLC (US) 2010-09-21 US disclosed
US-20060079543-A1 Anilino-pyrimidine analogs WYETH (US) 2006-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079543-A1 Anilino-pyrimidine analogs DPYD, TYMP, ADORA3 IKBKB 3246/4885CDK2 11/4885CDK4 69/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.