SCHEMBL3517140

SCHEMBL3517140

Nc1ncnc2c1nc(Br)n2CCC1CCNCC1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.60
HSP90AB1 P08238 3/20 0.60
ADORA2A P29274 16/20 0.59
ADORA1 P30542 16/20 0.59
ADORA2B P29275 12/20 0.59
ADORA3 P0DMS8 7/20 0.56
FBP1 P09467 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4954196 0.88 ADORA2A (0.61) HSP90AA1HSP90AB1ADORA2AADORA1ADORA2B
SCHEMBL13731182 0.82 ADORA2A (0.58) HSP90AA1HSP90AB1ADORA2AADORA1ADORA2B
SCHEMBL3746480 0.81 HSP90AA1 (0.63) HSP90AA1HSP90AB1ADORA2AADORA1ADORA2B
SCHEMBL3515942 0.81 ADORA2A (0.56) HSP90AA1HSP90AB1ADORA2AADORA1ADORA2B
SCHEMBL3111832 0.80 HSP90AA1 (0.63) HSP90AA1HSP90AB1ADORA2AADORA1ADORA2B
SCHEMBL13845675 0.78 HSP90AA1 (0.77) HSP90AA1HSP90AB1
SCHEMBL27774220 0.77 HSP90AA1 (0.52) HSP90AA1HSP90AB1ADORA2AADORA1ADORA2B
SCHEMBL3517082 0.77 HSP90AA1 (0.76) HSP90AA1HSP90AB1
SCHEMBL3516432 0.76 ADORA2A (0.56) ADORA2AADORA1ADORA2B
SCHEMBL3119723 0.76 HSP90AA1 (1.00) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2219448-A1 THERAPEUTIC COMPOUNDS AND THEIR USE IN TREATING DISEASES AND DISORDERS Myriad Pharmaceuticals, Inc. (US) 2010-08-25 EP disclosed
WO-2009065035-A1 THERAPEUTIC COMPOUNDS AND THEIR USE IN TREATING DISEASES AND DISORDERS MYRIAD GENETICS, INC. (US) 2009-05-22 WO disclosed
WO-2009065035-A1 THERAPEUTIC COMPOUNDS AND THEIR USE IN TREATING DISEASES AND DISORDERS MYRIAD GENETICS, INC. (US) 2009-05-22 WO disclosed