Furofenac

Furofenac

SCHEMBL35188

CCC1Cc2cc(CC(=O)O)ccc2O1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 1/20 0.46
POLB P06746 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
FFAR1 O14842 2/20 0.42
TDP1 Q9NUW8 2/20 0.41
AKR1B1 P15121 3/20 0.41
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.39
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
RGS12 O14924 1/20 0.39
LMNA P02545 1/20 0.39
NFKB1 P19838 1/20 0.39
APEX1 P27695 1/20 0.39
THPO P40225 1/20 0.39
BLM P54132 1/20 0.39
GNAI1 P63096 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Furofenac SCHEMBL29413089 1.00 TBXA2R (0.46) TBXA2RPOLBL3MBTL1FFAR1TDP1
SCHEMBL10388108 0.87 TBXA2R (0.46) TBXA2RPOLBL3MBTL1FFAR1TDP1
SCHEMBL13085688 0.82 TDP1 (0.61) TBXA2RPOLBL3MBTL1FFAR1TDP1
SCHEMBL14457195 0.80 FFAR1 (0.42) TBXA2RPOLBFFAR1TDP1AKR1B1
Tiopinac SCHEMBL9709495 0.80 AKR1B1 (0.69) AKR1B1HRH1
SCHEMBL16742113 0.79 TDP1 (0.66) POLBTDP1AKR1B1TSHRALDH1A1
SCHEMBL9443900 0.79 HRH3 (0.40) TBXA2RPOLBFFAR1TDP1ALDH1A1
SCHEMBL11373080 0.77 TDP1 (0.51) POLBFFAR1TDP1AKR1B1ALDH1A1
SCHEMBL9443905 0.76 FFAR1 (0.40) TBXA2RFFAR1CYP4F2CYP4A11MEN1
SCHEMBL5536590 0.75 HRH3 (0.41) TBXA2RPOLBFFAR1TDP1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6802 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE50218-E1 Non-steroidal anti-inflammatory ophthalmic compositions SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2024-11-26 US claimed
CN-118141602-A Lacrimal canaliculus embolism 上海曙瑞科技有限公司 2024-06-07 CN claimed
EP-4308063-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORM Procaps SA (US) 2024-01-24 EP claimed
EP-4185277-A1 SOFT SHELL GELATIN CAPSULES Procaps SA (US) 2023-05-31 EP claimed
WO-2023075715-A1 A PHARMACEUTICAL FORMULATION INCLUDING LEUKOTRIENE RECEPTOR ANTAGONISTS AND/OR LEUKOTRIENE SYNTHESIS INHIBITORS COMBINED WITH NON-STEROIDAL ANTI-INFLAMMATORY DRUGS (NSAIDS) VSY BIYOTEKNOLOJI VE ILAC SANAYI ANONIM SIRKETI (TR) 2023-05-04 WO claimed
US-20230088240-A1 ACCELERATING THE DRYING RATE OF SOFTGEL CAPSULES GLAS AMERICAS LLC 2023-03-23 US claimed
WO-2022197983-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORM PROCAPS SA (US) 2022-09-22 WO claimed
US-20220296529-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORMS WITHIN SAID CAPSULES GLAS AMERICAS LLC 2022-09-22 US claimed
EP-3998932-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS Parsons, C. Lowell (US) 2022-05-25 EP claimed
US-11273162-B2 Compositions and methods targeting HCN channels for breathing therapeutics MISSISSIPPI STATE UNIVERSITY (US) 2022-03-15 US claimed
EP-0167566-A4 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME. SUNSHINE ABRAHAM (US) 1987-06-29 EP claimed
EP-0205492-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE, Abraham (US) 1986-12-30 EP claimed
WO-1986003681-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE ABRAHAM 1986-07-03 WO claimed
EP-0167566-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE, Abraham (US) 1986-01-15 EP claimed
WO-1985003443-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING DIPHENHYDRAMINE AND METHODS OF USING SAME RICHARDSON-VICKS, INC. (US) 1985-08-15 WO claimed
WO-1985002542-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE ABRAHAM 1985-06-20 WO claimed
EP-0114886-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE. SUNSHINE ABRAHAM (US) 1984-08-08 EP claimed
WO-1984000490-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE AND METHODS OF USING SAME SUNSHINE ABRAHAM 1984-02-16 WO claimed
EP-0008752-B1 PROCESS FOR THE PREPARATION OF 2,3-DIHYDRO-2-ETHYL-BENZOFURAN-5-ACETIC ACID ALFA FARMACEUTICI S.p.A. (IT) 1981-08-12 EP claimed
EP-0008752-A1 Process for the preparation of 2,3-dihydro-2-ethyl-benzofuran-5-acetic acid ALFA FARMACEUTICI S.p.A. (IT) 1980-03-19 EP claimed