SCHEMBL3537474

SCHEMBL3537474

O=C(O)N1CCN(c2cc(-c3ccccc3F)ncn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.52
CYP1A2 P05177 5/20 0.50
CYP2C19 P33261 3/20 0.49
DPP4 P27487 3/20 0.49
ALOX15 P16050 1/20 0.49
HRH4 Q9H3N8 1/20 0.47
TSHR P16473 2/20 0.46
NPC1 O15118 2/20 0.46
RECQL P46063 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
TAF1 P21675 1/20 0.41
CECR2 Q9BXF3 1/20 0.41
BRD9 Q9H8M2 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
TACR3 P29371 1/20 0.41
KDM4E B2RXH2 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268033 0.83 SMARCA2 (0.53) FAAHCYP1A2CYP2C19DPP4ALOX15
SCHEMBL3535125 0.81 FAAH (0.47) FAAHCYP1A2CYP2C19DPP4ALOX15
SCHEMBL12991226 0.81 FAAH (0.47) FAAHCYP1A2CYP2C19DPP4ALOX15
SCHEMBL12991318 0.81 LRRK2 (0.49) FAAHCYP1A2CYP2C19DPP4ALOX15
SCHEMBL3274302 0.79 CYP1A2 (0.71) CYP1A2CYP2C19DPP4ALOX15HRH4
SCHEMBL3274064 0.79 FAAH (0.58) FAAHSMN1; SMN2ALDH1A1LMNALOXL2
SCHEMBL3275295 0.79 FAAH (0.83) FAAHLOXL2
SCHEMBL3528677 0.78 PIM1 (0.42) FAAHALOX15TSHRNPC1RAB9A
SCHEMBL3274898 0.77 FAAH (0.51) FAAHCYP1A2CYP2C19ALOX15TSHR
SCHEMBL3535103 0.75 FAAH (0.52) FAAHCYP1A2CYP2C19ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858786-B2 Pyrimidines and pyrazines useful as modulators of ion channels VERTEX PHARMACEUTICALS INCOROPATED (US) 2010-12-28 US disclosed
US-20070093454-A1 Pyrimidines and pyrazines useful as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED 2007-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070093454-A1 Pyrimidines and pyrazines useful as modulators of ion channels KCNJ1, KCNJ2, KCNJ11 FAAH 2875/4885CYP1A2 2596/4885CYP2C19 2702/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.