SCHEMBL354135

SCHEMBL354135

COc1ccc(CO[C@@H](C/C=C(\C)I)CCO)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.37
AGXT P21549 2/20 0.37
APP P05067 5/20 0.37
TBXAS1 P24557 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
SLC6A4 P31645 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
FFAR1 O14842 1/20 0.35
CALM1 P0DP23 1/20 0.35
AOC3 Q16853 1/20 0.34
HTT P42858 1/20 0.34
LDHA P00338 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353344 0.87 MEN1 (0.43) IDO1AGXTAPPTBXAS1CA1
SCHEMBL17305606 0.87 MEN1 (0.43) IDO1AGXTAPPTBXAS1CA1
SCHEMBL26512096 0.79 CA1 (0.45) IDO1AGXTAPPTBXAS1CA1
SCHEMBL7140177 0.74 TBXAS1 (0.43) IDO1AGXTTBXAS1CALM1
SCHEMBL13030081 0.74 TBXAS1 (0.43) IDO1AGXTTBXAS1CALM1
SCHEMBL7140172 0.74 TBXAS1 (0.43) IDO1AGXTTBXAS1CALM1
SCHEMBL26985881 0.73 CYP2C9 (0.53) IDO1AGXTAPPTBXAS1CA1
SCHEMBL12769997 0.72 SLC6A4 (0.49) IDO1AGXTAPPCA1CA2
SCHEMBL27032518 0.72 SLC6A4 (0.49) IDO1AGXTAPPCA1CA2
SCHEMBL27131530 0.72 SLC6A4 (0.49) IDO1AGXTAPPCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231590-B9 ANTITUMORAL COMPOUNDS PHARMA MAR SA (ES) 2012-08-15 EP disclosed
EP-2231590-B1 ANTITUMORAL COMPOUNDS PHARMA MAR SA (ES) 2012-03-14 EP disclosed