SCHEMBL3546146

SCHEMBL3546146

CC(CNC1=NCCN1)C(=O)N1CCC(C(=O)N[C@@H](CC(=O)O)c2cnc3ccccc3c2)CC1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.74
ITGA2B P08514 13/20 0.74
ITGAV P06756 13/20 0.74
ITGB5 P18084 3/20 0.74
F2R P25116 1/20 0.54
CAPN1 P07384 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13344622 0.86 ITGB3 (0.73) ITGB3ITGA2BITGAVITGB5
SCHEMBL3534624 0.85 ITGB3 (1.00) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL3533265 0.85 ITGB3 (0.78) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL13344586 0.80 ITGB3 (0.68) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL13344615 0.79 ITGB3 (0.85) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL13369229 0.76 ITGB3 (0.83) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL13344609 0.75 ITGB3 (0.82) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL13344619 0.75 ITGB3 (0.76) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL3539083 0.74 ITGB3 (0.77) ITGB3ITGA2BITGAVITGB5F2R
SCHEMBL13344577 0.73 ITGB3 (0.66) ITGB3ITGA2BITGAVITGB5F2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7718673-B2 Isonipecotamides for the treatment of integrin-mediated disorders ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2010-05-18 US claimed
US-7718673-B2 Isonipecotamides for the treatment of integrin-mediated disorders ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2010-05-18 US disclosed