SCHEMBL3562428

SCHEMBL3562428

CCCn1c(C)c(C(=O)Nc2ccc(Oc3cc(NC(=O)N4CCC(C)CC4)ncn3)c(F)c2)c(=O)n1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.56
KDR P35968 18/20 0.56
IGF1R P08069 15/20 0.56
MST1R Q04912 2/20 0.46
AURKA O14965 1/20 0.45
JAK2 O60674 1/20 0.45
RPS6KA5 O75582 1/20 0.45
ABL1 P00519 1/20 0.45
INSR P06213 1/20 0.45
LCK P06239 1/20 0.45
RET P07949 1/20 0.45
KIT P10721 1/20 0.45
PIM1 P11309 1/20 0.45
FGFR1 P11362 1/20 0.45
SRC P12931 1/20 0.45
PRKACA P17612 1/20 0.45
RPS6KB1 P23443 1/20 0.45
JAK1 P23458 1/20 0.45
MAPK3 P27361 1/20 0.45
AKT1 P31749 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL198531 0.93 KDR (0.58) METKDRIGF1RMST1RAURKA
SCHEMBL200162 0.93 MET (0.58) METKDRIGF1RMST1RINSR
SCHEMBL197608 0.93 KDR (0.58) METKDRIGF1RMST1RAURKA
SCHEMBL200732 0.92 MET (0.56) METKDRIGF1RMST1RAURKA
SCHEMBL199596 0.91 MET (0.53) METKDRIGF1RMST1RAURKA
SCHEMBL199595 0.91 MET (0.53) METKDRIGF1RMST1RAURKA
SCHEMBL14003861 0.85 KDR (0.53) METKDRIGF1RMST1RAURKA
SCHEMBL2742559 0.84 MET (0.61) METKDRIGF1RMST1RAURKA
SCHEMBL198021 0.84 KDR (0.59) METKDRIGF1RMST1R
SCHEMBL200073 0.83 MET (0.66) METKDRIGF1RMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858623-B2 Substituted amide derivatives and methods of use AMGEN INC. (US) 2010-12-28 US claimed