SCHEMBL3565795

SCHEMBL3565795

Cc1ccc(C(=O)CC2c3nc(-c4ccncn4)cc(=O)n3CNC2(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.40
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3572719 0.92 GSK3B (0.42) GSK3BCYP2D6
SCHEMBL3575939 0.92 GSK3B (0.42) GSK3BCYP2D6
SCHEMBL3567458 0.92 GSK3B (0.43) GSK3BCYP2D6
SCHEMBL3579597 0.90 GSK3B (0.43) GSK3BCYP3A4CYP2D6
SCHEMBL3570867 0.89 GSK3B (0.39) GSK3BCYP2D6
SCHEMBL3578451 0.89 GSK3B (0.41) GSK3BCYP2D6
SCHEMBL3564980 0.85 GSK3B (0.45) GSK3BCYP3A4CYP2D6
SCHEMBL3579567 0.84 GSK3B (0.41) GSK3BCYP3A4CYP2D6
SCHEMBL3568702 0.82 CYP3A4 (0.40) GSK3BCYP3A4CYP2D6
SCHEMBL3564702 0.78 GSK3B (0.42) GSK3BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781440-B2 Use of substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives SANOFI-AVENTIS (FR) 2010-08-24 US claimed