SCHEMBL3575939

SCHEMBL3575939

CC1(C)NCn2c(nc(-c3ccncn3)cc2=O)C1CC(=O)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.42
CYP2D6 P10635 4/20 0.40
CYP1A2 P05177 2/20 0.40
CSNK1A1 P48729 1/20 0.40
GSK3A P49840 1/20 0.40
GRM1 Q13255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3565795 0.92 GSK3B (0.40) GSK3BCYP2D6
SCHEMBL3572719 0.91 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3567458 0.91 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3579597 0.90 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3570867 0.88 GSK3B (0.39) GSK3BCYP2D6
SCHEMBL3578451 0.88 GSK3B (0.41) GSK3BCYP2D6CYP1A2
SCHEMBL3566582 0.85 GSK3B (0.42) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL3564980 0.84 GSK3B (0.45) GSK3BCYP2D6CYP1A2GSK3A
SCHEMBL3568702 0.80 CYP3A4 (0.40) GSK3BCYP2D6CYP1A2
SCHEMBL3578475 0.79 GSK3B (0.44) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781440-B2 Use of substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives SANOFI-AVENTIS (FR) 2010-08-24 US claimed