Pyridine

Pyridine

SCHEMBL3566017

Cc1cnc(NC2CCCC(C)C2C)nc1CC#N.c1ccncc1

nearest known ligand 0.33

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 4/20 0.33
STAT3 P40763 4/20 0.33
JAK1 P23458 2/20 0.33
TYK2 P29597 2/20 0.33
JAK3 P52333 2/20 0.33
SYK P43405 2/20 0.32
MAPK1 P28482 1/20 0.32
ABL1 P00519 3/20 0.31
KDR P35968 3/20 0.31
GSK3B P49841 3/20 0.31
AURKB Q96GD4 3/20 0.31
GBA1 P04062 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30
LATS1 O95835 3/20 0.30
LATS2 Q9NRM7 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL3574027 0.83 JAK2 (0.42) JAK2STAT3JAK1TYK2JAK3
Pyridine SCHEMBL3562760 0.82 JAK2 (0.44) JAK2STAT3JAK1TYK2JAK3
Pyridine SCHEMBL3571503 0.82 CTSK (0.43) JAK2STAT3JAK1TYK2JAK3
Pyridine SCHEMBL5622345 0.81 MAPK1 (0.34) MAPK1GBA1TAS1R3TAS1R1LATS1
Pyridine SCHEMBL3569024 0.76 MEN1 (0.38) GSK3BGBA1
Pyridine SCHEMBL3572010 0.71 JAK2 (0.33) JAK2STAT3JAK1TYK2JAK3
SCHEMBL3566014 0.71 SYK (0.32) SYKMAPK1TAS1R3TAS1R1
Pyridine SCHEMBL3573055 0.69 TYRO3 (0.37) JAK2STAT3JAK1TYK2JAK3
Pyridine SCHEMBL3569208 0.69 MAPT (0.37)
SCHEMBL7357712 0.68 GAA (0.47) JAK2MAPK1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7855212-B2 Pyridinyl acetonitriles MERCK SERONO SA (CH) 2010-12-21 US claimed
US-20070060594-A1 Pyridinyl acetonitriles APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (NL) 2007-03-15 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070060594-A1 Pyridinyl acetonitriles GSK3B, GSK3A, MAPK3 JAK2 432/4885STAT3 638/4885JAK1 296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.