SCHEMBL357407

SCHEMBL357407

COc1cc(C(=O)Oc2ccc(C(=O)O)cc2OC)ccc1O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.76
TSHR P16473 3/20 0.65
MAPT P10636 1/20 0.65
CA12 O43570 1/20 0.65
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA4 P22748 1/20 0.65
CA6 P23280 1/20 0.65
CA7 P43166 1/20 0.65
TPMT P51580 1/20 0.65
CA9 Q16790 1/20 0.65
CA14 Q9ULX7 1/20 0.65
KMT2A Q03164 3/20 0.58
HDAC6 Q9UBN7 1/20 0.58
RAB9A P51151 3/20 0.58
MEN1 O00255 2/20 0.58
SLC22A6 Q4U2R8 1/20 0.58
SLC22A8 Q8TCC7 1/20 0.58
HSD17B2 P37059 1/20 0.57
KDM4E B2RXH2 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6213459 0.93 HTT (0.64) HTTTSHRMAPTCA12CA1
SCHEMBL27620944 0.89 MAPT (0.67) HTTTSHRMAPTCA12CA1
SCHEMBL2791210 0.89 MAPT (0.82) HTTTSHRMAPTCA12CA1
SCHEMBL21114354 0.88 CA12 (0.69) HTTTSHRMAPTCA12CA1
Vanillic Acid SCHEMBL9711598 0.87 HTT (1.00) HTTTSHRMAPTCA12CA1
Vanillic Acid SCHEMBL26179 0.87 HTT (1.00) HTTTSHRMAPTCA12CA1
Vanillic Acid SCHEMBL29378740 0.87 HTT (1.00) HTTTSHRMAPTCA12CA1
Vanillic Acid SCHEMBL6697041 0.85 HTT (0.96) HTTTSHRCA12CA1CA2
Vanillic Acid SCHEMBL17443329 0.85 HTT (0.96) HTTTSHRCA12CA1CA2
Vanillic Acid SCHEMBL18334646 0.85 HTT (0.96) HTTTSHRCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011067571-A1 CO - CRYSTALS OF A TRIAZOLO [4,5 - D] PYRIMIDINE PLATELET AGGREGATION INHIBITOR ASTRAZENECA AB (SE) 2011-06-09 WO claimed
US-20120014883-A1 Compositions Comprising Derivatives Of Essential Oil Compounds And Use In Personal Care Products THE PROCTER & GAMBLE COMPANY 2012-01-19 US disclosed
US-20110288161-A1 METHODS FOR TREATMENT OF THIOL-CONTAINING COMPOUND DEFICIENT CONDITIONS NATIONAL JEWISH MEDICAL AND RESEARCH CENTER 2011-11-24 US disclosed
EP-2383330-A1 A stabilized liquid enzyme composition Novozymes A/S (DK) 2011-11-02 EP disclosed
WO-2011067571-A1 CO - CRYSTALS OF A TRIAZOLO [4,5 - D] PYRIMIDINE PLATELET AGGREGATION INHIBITOR ASTRAZENECA AB (SE) 2011-06-09 WO disclosed
WO-2011067571-A1 CO - CRYSTALS OF A TRIAZOLO [4,5 - D] PYRIMIDINE PLATELET AGGREGATION INHIBITOR ASTRAZENECA AB (SE) 2011-06-09 WO disclosed
WO-2011064237-A1 CRYSTALLINE FORMS OF SUBSTITUTED PYRAZOLOPYRIMIDINES MERZ PHARMA GMBH & CO. KGAA (DE) 2011-06-03 WO disclosed
US-20110104305-A1 COMPOUNDS AND METHODS FOR THIOL-CONTAINING COMPOUND EFFLUX AND CANCER TREATMENT DAY BRIAN J 2011-05-05 US disclosed
WO-1992017550-A1 BIODEGRADABLE AZO DYES IDAHO RESEARCH FOUNDATION, INC. (US) 1992-10-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288161-A1 METHODS FOR TREATMENT OF THIOL-CONTAINING COMPOUND DEFICIENT CONDITIONS ABCC1, SLC47A2, SLC47A1 HTT 987/4885TSHR 4043/4885MAPT 3843/4885
US-20110104305-A1 COMPOUNDS AND METHODS FOR THIOL-CONTAINING COMPOUND EFFLUX AND CANCER TREATMENT ABCC1, ABCC2, ABCB1 HTT 2358/4885TSHR 3356/4885MAPT 4577/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.