SCHEMBL3578489

SCHEMBL3578489

NC(=O)c1cccc2nc(-c3ccc(OCCN4CCCC4)cc3)[nH]c12

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.71
DHODH Q02127 1/20 0.71
CHEK2 O96017 2/20 0.64
ACHE P22303 6/20 0.64
ADORA3 P0DMS8 1/20 0.55
ADORA2A P29274 1/20 0.55
ADORA2B P29275 1/20 0.55
ADORA1 P30542 1/20 0.55
TBK1 Q9UHD2 4/20 0.54
CDK2 P24941 1/20 0.53
IKBKE Q14164 1/20 0.53
AURKB Q96GD4 1/20 0.53
CHEK1 O14757 1/20 0.51
GCGR P47871 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6810424 0.86 PARP1 (0.57) PARP1DHODHCHEK2ACHEADORA2A
SCHEMBL3578485 0.85 PARP1 (0.96) PARP1DHODHCHEK2ACHEAURKB
SCHEMBL7135402 0.83 PARP1 (0.58) PARP1DHODHCHEK2ACHEAURKB
SCHEMBL6800865 0.82 PARP1 (0.52) PARP1DHODHCHEK2ACHEADORA2A
SCHEMBL6029990 0.82 PARP1 (0.60) PARP1DHODHCHEK2ACHECHEK1
SCHEMBL6806306 0.80 PARP1 (0.47) PARP1DHODHCHEK2ACHETBK1
SCHEMBL3575241 0.80 MAP4K4 (0.72) PARP1DHODHCHEK2ACHEADORA3
SCHEMBL6810662 0.79 PARP1 (0.49) PARP1DHODHCHEK2ACHEADORA2A
SCHEMBL3575819 0.79 CHEK1 (0.65) PARP1DHODHCHEK2ACHEADORA3
SCHEMBL6805060 0.79 AURKB (0.53) PARP1DHODHCHEK2TBK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed