SCHEMBL3581228

SCHEMBL3581228

NC(=O)c1ccc(C(=O)c2ccc3c(c2)CC(=O)N3)cc1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 16/20 0.55
HDAC3 O15379 1/20 0.49
AHR P35869 1/20 0.49
EPHX2 P34913 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29567045 0.91 SMYD3 (0.57) SMYD3HDAC3AHREPHX2
SCHEMBL3190474 0.91 SMYD3 (0.57) SMYD3HDAC3AHREPHX2
SCHEMBL3575509 0.90 SMYD3 (0.52) SMYD3HDAC3AHREPHX2
SCHEMBL3573876 0.89 SMYD3 (0.56) SMYD3HDAC3AHR
Hydrochloric Acid SCHEMBL28849276 0.89 SMYD3 (0.56) SMYD3HDAC3AHREPHX2
SCHEMBL3569829 0.88 SMYD3 (0.55) SMYD3HDAC3AHREPHX2
SCHEMBL3255662 0.86 SMYD3 (0.53) SMYD3AHREPHX2
SCHEMBL11461325 0.85 AHR (0.66) SMYD3HDAC3AHREPHX2
SCHEMBL16180358 0.84 PDE3B (0.61) SMYD3HDAC3AHREPHX2
SCHEMBL14565018 0.81 SMYD3 (0.50) SMYD3HDAC3AHREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7749530-B2 Kinase inhibitors ALLERGAN, INC. (US) 2010-07-06 US disclosed
WO-2010075197-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2010-07-01 WO disclosed
US-7692005-B2 Kinase inhibitors ALLERGAN, INC. (US) 2010-04-06 US disclosed
US-20090208557-A1 Kinase inhibitors ALLERGAN, INC. 2009-08-20 US disclosed
EP-1902025-A1 KINASE INHIBITORS Allergan, Inc. (US) 2008-03-26 EP disclosed
US-20070032478-A1 Kinase Inhibitors ALLERGAN, INC. 2007-02-08 US disclosed
WO-2007008895-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2007-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090208557-A1 Kinase inhibitors PTK2, MAP3K6, MAP3K20 SMYD3 3186/4885HDAC3 1826/4885AHR 2818/4885
US-20070032478-A1 Kinase Inhibitors ABL1, LCK, ERBB2 SMYD3 1968/4885HDAC3 3313/4885AHR 2478/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.