SCHEMBL3583587

SCHEMBL3583587

CCOC(=O)c1cc(-c2cc(O)c(O)c([N+](=O)[O-])c2)n(CC)c1-c1ccc(C(F)(F)F)nc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
HPGD P15428 2/20 0.38
CHRNA7 P36544 5/20 0.37
CA9 Q16790 1/20 0.35
GAA P10253 3/20 0.34
MAPT P10636 2/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
POLB P06746 1/20 0.34
CSNK1D P48730 1/20 0.34
ALOX5 P09917 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28780430 0.90 TTR (0.35)
SCHEMBL1446798 0.85 ALDH1A1 (0.36) ALDH1A1HPGDCHRNA7GAAMAPT
SCHEMBL3587861 0.76 MAPT (0.38) ALDH1A1HPGDGAAMAPTHTT
SCHEMBL3584510 0.75 ALDH1A1 (0.36) ALDH1A1HPGDMAPTPOLB
SCHEMBL3587266 0.75 ALDH1A1 (0.38) ALDH1A1HPGDMAPTNPSR1POLB
SCHEMBL3591011 0.74 TTR (0.39) ALDH1A1HPGDCA9MAPTPTGS1
SCHEMBL1446969 0.73 ALDH1A1 (0.36) ALDH1A1HPGDCHRNA7MAPTNPSR1
SCHEMBL1446919 0.72 MAPT (0.36) ALDH1A1HPGDGAAMAPTHTT
SCHEMBL3586613 0.71 ALDH1A1 (0.44) ALDH1A1HPGDGAAMAPTHTT
SCHEMBL25011698 0.71 MAPT (0.43) ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9446012-B2 Pharmaceutical compounds BIAL—PORTELA & CA, S.A. (PT) 2016-09-20 US disclosed
US-20140024682-A1 PHARMACEUTICAL COMPOUNDS BIAL - PORTELA & CA, S.A. (PT) 2014-01-23 US disclosed
US-8536203-B2 Pharmaceutical compounds BIAL-PORTELA & CA, S.A. (PT) 2013-09-17 US disclosed
EP-2617713-A1 New Pharmaceutical Compounds BIAL - Portela & Ca., S.A. (PT) 2013-07-24 EP disclosed
US-20100168113-A1 Pharmaceutical Compounds BIAL-PORTELA & CA., S.A. (PT) 2010-07-01 US disclosed
CN-101248064-A Nitrocatechol derivatives as COMT inhibitors PORTELA & CA SA (PT) 2008-08-20 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168113-A1 Pharmaceutical Compounds PMP22, CNR2, OPRL1 ALDH1A1 1070/4885HPGD 307/4885CHRNA7 187/4885
US-20140024682-A1 PHARMACEUTICAL COMPOUNDS PMP22, CNR2, OPRL1 ALDH1A1 1070/4885HPGD 307/4885CHRNA7 187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.