SCHEMBL3584828

SCHEMBL3584828

CC(C)(O)Cn1ccc2c(N)cccc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.58
KDM4E B2RXH2 7/20 0.39
ALDH1A1 P00352 5/20 0.38
HPGD P15428 2/20 0.38
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TTR P02766 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
NSD2 O96028 2/20 0.37
DHPS P49366 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
GRM2 Q14416 4/20 0.36
JAK2 O60674 1/20 0.36
ELANE P08246 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17577600 0.84 KDM4E (0.40) PARP1KDM4EALDH1A1HPGDTSHR
SCHEMBL9394351 0.80 PARP1 (0.61) PARP1KDM4EALDH1A1HPGDTSHR
SCHEMBL12702816 0.77 PARP1 (0.67) PARP1GRM2
SCHEMBL17577713 0.77 KDM4E (0.56) KDM4EALDH1A1TDP1SMN1; SMN2
SCHEMBL1896689 0.77 PARP1 (0.71) PARP1KDM4EALDH1A1HPGDTSHR
SCHEMBL3576491 0.77 PARP1 (0.58) PARP1KDM4EALDH1A1HPGDTSHR
SCHEMBL1590065 0.76 PARP1 (0.65) PARP1KDM4EALDH1A1HPGDTSHR
SCHEMBL4147543 0.74 PARP1 (0.62) PARP1KDM4EALDH1A1NSD2DHPS
SCHEMBL3753520 0.73 PARP1 (0.62) PARP1ALDH1A1HPGDTSHRCYP3A4
SCHEMBL3747700 0.73 PARP1 (0.62) PARP1ALDH1A1HPGDTSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816371-B2 Bicycloheteroaryl compounds as P2X7 modulators and uses thereof RENOVIS, INC. (US) 2010-10-19 US claimed