SCHEMBL3576491

SCHEMBL3576491

CC(O)Cn1ccc2c(N)cccc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.58
KDM4E B2RXH2 6/20 0.44
HTR2C P28335 4/20 0.39
HTR2A P28223 3/20 0.39
ALDH1A1 P00352 5/20 0.38
TSHR P16473 3/20 0.38
HSD17B10 Q99714 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
HPGD P15428 2/20 0.38
CYP3A4 P08684 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ELANE P08246 1/20 0.38
DHPS P49366 1/20 0.37
PSMB1 P20618 1/20 0.37
PSMB5 P28074 1/20 0.37
GRM2 Q14416 2/20 0.36
NPC1 O15118 1/20 0.36
RORA P35398 1/20 0.36
NR5A1 Q13285 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17577751 0.84 HTR2A (0.50) PARP1KDM4EHTR2CHTR2AALDH1A1
SCHEMBL9394351 0.80 PARP1 (0.61) PARP1KDM4EALDH1A1TSHRHSD17B10
SCHEMBL1896689 0.77 PARP1 (0.71) PARP1KDM4EALDH1A1TSHRHSD17B10
SCHEMBL12702816 0.77 PARP1 (0.67) PARP1GRM2
SCHEMBL3584828 0.77 PARP1 (0.58) PARP1KDM4EALDH1A1TSHRHSD17B10
SCHEMBL1590065 0.76 PARP1 (0.65) PARP1KDM4EALDH1A1TSHRHSD17B10
SCHEMBL4147543 0.74 PARP1 (0.62) PARP1KDM4EALDH1A1DHPSGRM2
SCHEMBL3746261 0.73 PARP1 (0.62) PARP1ALDH1A1GRM2
SCHEMBL3753520 0.73 PARP1 (0.62) PARP1ALDH1A1TSHRHSD17B10TDP1
SCHEMBL13243839 0.73 P2RX7 (0.49) PARP1KDM4EHTR2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816371-B2 Bicycloheteroaryl compounds as P2X7 modulators and uses thereof RENOVIS, INC. (US) 2010-10-19 US claimed