SCHEMBL358735

SCHEMBL358735

Cc1c2cccc(C(N)=O)c2nn1C1CCCNC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.49
RPS6KB1 P23443 6/20 0.49
AURKA O14965 5/20 0.49
PARP2 Q9UGN5 4/20 0.48
PARP3 Q9Y6F1 3/20 0.48
DYRK1A Q13627 2/20 0.48
TNKS O95271 1/20 0.48
CHRM2 P08172 1/20 0.48
CHRM1 P11229 1/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
ADRA1A P35348 1/20 0.48
SLC6A3 Q01959 1/20 0.48
KCNH2 Q12809 1/20 0.48
PARP15 Q460N3 1/20 0.48
PARP14 Q460N5 1/20 0.48
PARP10 Q53GL7 1/20 0.48
PARP12 Q9H0J9 1/20 0.48
TNKS2 Q9H2K2 1/20 0.48
PARP4 Q9UKK3 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL358621 0.93 RPS6KB1 (0.47) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL12503295 0.90 PARP1 (0.47) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL359270 0.87 PARP1 (0.49) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL359581 0.86 RPS6KB1 (0.48) PARP1RPS6KB1AURKAPARP2
SCHEMBL359970 0.85 RPS6KB1 (0.48) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL358870 0.84 F10 (0.38) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL12503212 0.83 PARP1 (0.41) PARP1RPS6KB1AURKAPARP2SLC6A2
SCHEMBL359495 0.82 PARP1 (0.46) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL359319 0.81 RPS6KB1 (0.45) PARP1RPS6KB1AURKAPARP2PARP3
SCHEMBL359540 0.81 RAD52 (0.44) PARP1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO claimed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed