SCHEMBL358870

SCHEMBL358870

Cc1c2cccc(C(=O)NN(C)C)c2nn1C1CCCNC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.38
AURKA O14965 3/20 0.37
RPS6KB1 P23443 3/20 0.37
PARP1 P09874 7/20 0.37
HTR6 P50406 3/20 0.36
PARP2 Q9UGN5 3/20 0.34
PARP3 Q9Y6F1 3/20 0.34
TNKS O95271 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
ADRA1A P35348 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
DYRK1A Q13627 1/20 0.34
PARP15 Q460N3 1/20 0.34
PARP14 Q460N5 1/20 0.34
PARP10 Q53GL7 1/20 0.34
PARP12 Q9H0J9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL359217 0.94 RPS6KB1 (0.35) F10AURKARPS6KB1PARP1HTR6
SCHEMBL357860 0.88 NR3C1 (0.36) AURKARPS6KB1PARP1PARP2HTR3A
SCHEMBL359540 0.87 RAD52 (0.44) F10PARP1KCNH2
SCHEMBL12503295 0.85 PARP1 (0.47) F10AURKARPS6KB1PARP1HTR6
SCHEMBL358735 0.84 PARP1 (0.49) AURKARPS6KB1PARP1PARP2PARP3
SCHEMBL358998 0.84 SCN4A (0.34) AURKARPS6KB1PARP1PARP2PARP3
SCHEMBL359667 0.83 RPS6KB1 (0.34) AURKARPS6KB1PARP1CHRM2CHRM1
SCHEMBL359562 0.81 PARP1 (0.32) PARP1HTR3A
SCHEMBL358798 0.80 RAD52 (0.46) PARP1KCNH2
SCHEMBL12503212 0.79 PARP1 (0.41) AURKARPS6KB1PARP1HTR6PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO claimed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed