SCHEMBL3588047

SCHEMBL3588047

O=C(Cn1ccc2cc(-c3ccc(F)cc3)ccc21)NCCNCC1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 8/20 0.52
NPY5R Q15761 2/20 0.46
FAAH O00519 1/20 0.44
NTSR1 P30989 1/20 0.42
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3600291 0.92 GRIN2B (0.55) GRIN2BNPY5RPOLBRAB9ASMN1; SMN2
SCHEMBL3596258 0.90 NPC1 (0.47) GRIN2BNPY5RFAAHNTSR1RAB9A
SCHEMBL3602171 0.84 KDM4E (0.43) GRIN2BNPY5RFAAHNTSR1POLB
SCHEMBL3600784 0.84 GRIN2B (0.48) GRIN2BNPY5RNTSR1POLB
SCHEMBL3598451 0.83 ALDH1A1 (0.45) GRIN2BNTSR1POLBSMN1; SMN2
SCHEMBL3601361 0.82 KDM4E (0.44) GRIN2BNPY5RFAAHPOLBSMN1; SMN2
SCHEMBL3597368 0.82 TSHR (0.46) GRIN2BNPY5RPOLBRAB9A
SCHEMBL3602467 0.82 KDM4E (0.46) GRIN2BNPY5RPOLBRAB9ASMN1; SMN2
SCHEMBL3644326 0.82 KDM4E (0.48) GRIN2BPOLBSMN1; SMN2
SCHEMBL3600113 0.82 GRIN2B (0.44) GRIN2BNPY5RPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
WO-2007115231-A2 CXCR4 MODULATORS CHEMOCENTRYX, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275965-A1 CXCR4 modulators CXCL12, CXCR4, CXCR1 GRIN2B 2950/4885NPY5R 4199/4885FAAH 3521/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.