SCHEMBL359175

SCHEMBL359175

C=[C]c1ccc2ncccc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.57
POLB P06746 3/20 0.57
RAB9A P51151 2/20 0.57
ALDH1A1 P00352 4/20 0.53
MAPT P10636 3/20 0.53
ATM Q13315 2/20 0.53
HTT P42858 2/20 0.53
CASP1 P29466 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KDM4E B2RXH2 1/20 0.53
TP53 P04637 1/20 0.53
HSP90AA1 P07900 1/20 0.53
HSP90AB1 P08238 1/20 0.53
TSHR P16473 1/20 0.53
HSD17B10 Q99714 1/20 0.53
DYRK1A Q13627 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
CASP3 P42574 1/20 0.44
SENP7 Q9BQF6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851890 0.81 NPC1 (0.53) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL29843637 0.81 POLB (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL506632 0.81 POLB (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL31588535 0.81 POLB (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL2009640 0.81 NPC1 (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL738379 0.81 NPC1 (0.57) NPC1POLBRAB9AALDH1A1MAPT
SCHEMBL28153180 0.79 POLB (0.55) NPC1POLBRAB9AALDH1A1MAPT
Hydrochloric Acid SCHEMBL21436092 0.79 NPC1 (0.55) NPC1POLBRAB9AALDH1A1MAPT
Fluoride SCHEMBL28218511 0.79 POLB (0.55) NPC1POLBRAB9AALDH1A1MAPT
Quinoline SCHEMBL28269682 0.77 ALDH1A1 (0.59) NPC1POLBRAB9AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593107-A1 TYROSINE KINASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-22 EP disclosed
WO-2012009194-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed