SCHEMBL3604536

SCHEMBL3604536

CS(=O)(=O)NC(=O)OCC1CCCN(c2ccc(C#N)c3ccccc23)C1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AR P10275 13/20 0.47
DPP4 P27487 1/20 0.40
BCHE P06276 2/20 0.39
ACHE P22303 1/20 0.39
MAOB P27338 1/20 0.39
RPS6KB1 P23443 1/20 0.38
AKT1 P31749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3593053 0.83 AR (0.53) ARDPP4RPS6KB1AKT1
SCHEMBL4880027 0.79 AR (0.53) ARDPP4RPS6KB1AKT1
SCHEMBL4723950 0.79 AR (0.48) ARDPP4
SCHEMBL4871504 0.79 AR (0.50) AR
SCHEMBL27714512 0.78 AR (0.56) ARRPS6KB1AKT1
SCHEMBL3599646 0.78 AR (0.62) AR
SCHEMBL3615730 0.78 AR (0.62) AR
SCHEMBL3610108 0.78 AR (0.62) AR
Hydrochloric Acid SCHEMBL4881079 0.77 AR (0.55) ARRPS6KB1AKT1
Hydrochloric Acid SCHEMBL3604641 0.77 AR (0.60) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1553074-B1 FUSED BENZENE DERIVATIVE AND USE TAKEDA PHARMACEUTICAL (JP) 2014-06-18 EP disclosed
US-7649001-B2 Fused benzene derivative and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-01-19 US disclosed
EP-1553074-A1 FUSED BENZENE DERIVATIVE AND USE Takeda Pharmaceutical Company Limited (JP) 2005-07-13 EP disclosed