SCHEMBL3606408

SCHEMBL3606408

NCc1ccc(-c2cccnc2)o1.c1cncc(-c2ccc(CNCc3ccc(-c4cccnc4)o3)o2)c1

nearest known ligand 0.86

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 17/20 0.86
CYP2C19 P33261 15/20 0.83
CYP2D6 P10635 13/20 0.83
CYP2C9 P11712 13/20 0.83
CYP2B6 P20813 13/20 0.83
CYP2E1 P05181 12/20 0.83
CYP3A4 P08684 11/20 0.83
CYP1A2 P05177 6/20 0.61
SIGMAR1 Q99720 1/20 0.55
CYP2C8 P10632 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1791769 0.91 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL3608219 0.81 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL24700851 0.79 CYP2A6 (0.72) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL24701134 0.79 CYP2A6 (0.72) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL3604389 0.78 CYP2A6 (0.72) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL23789489 0.77 CYP2A6 (0.97) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL13035223 0.77 CYP2A6 (0.72) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
Hydrochloric Acid SCHEMBL23781570 0.76 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL3611340 0.75 CYP3A4 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6
SCHEMBL3617944 0.75 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8609708-B2 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2013-12-17 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
WO-2005066162-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2005-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP2C19 41/4885CYP2D6 7/4885
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP2C19 41/4885CYP2D6 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.