SCHEMBL3608219

SCHEMBL3608219

CNCc1ccc(-c2cccnc2)o1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 13/20 1.00
CYP2C19 P33261 9/20 1.00
CYP2D6 P10635 8/20 1.00
CYP2C9 P11712 8/20 1.00
CYP3A4 P08684 8/20 0.65
CYP2E1 P05181 6/20 0.65
CYP2B6 P20813 6/20 0.65
SOS1 Q07889 1/20 0.57
CD274 Q9NZQ7 1/20 0.53
EPHX2 P34913 1/20 0.51
PRMT6 Q96LA8 1/20 0.51
SIGMAR1 Q99720 1/20 0.49
CYP1A2 P05177 1/20 0.48
HRH1 P35367 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3606408 0.81 CYP2A6 (0.86) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL24701101 0.80 SOS1 (0.68) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL24700851 0.79 CYP2A6 (0.72) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL24701134 0.79 CYP2A6 (0.72) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL1791769 0.79 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL3611340 0.79 CYP3A4 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL3617944 0.79 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL3611062 0.78 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL13073854 0.78 CYP2A6 (0.65) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4
SCHEMBL3604825 0.78 CYP2A6 (1.00) CYP2A6CYP2C19CYP2D6CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8609708-B2 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2013-12-17 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
WO-2005066162-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2005-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP2C19 41/4885CYP2D6 7/4885
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP2C19 41/4885CYP2D6 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.