SCHEMBL3607722

SCHEMBL3607722

O=C(O)NCC#Cc1cccnc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 5/20 0.64
CHRNA4 P43681 5/20 0.64
CYP2A6 P11509 5/20 0.64
CYP2C9 P11712 3/20 0.64
CYP2B6 P20813 3/20 0.64
CYP2C19 P33261 3/20 0.64
CYP2D6 P10635 3/20 0.54
CYP2E1 P05181 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP1A2 P05177 2/20 0.53
CYP2C8 P10632 1/20 0.53
FFAR1 O14842 1/20 0.50
GRM5 P41594 5/20 0.46
PLOD2 O00469 1/20 0.45
PTGES O14684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13212066 0.83 CYP2A6 (0.55) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL13073855 0.80 PTPN11 (0.55) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL21591503 0.80 GRM5 (0.43) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL23781601 0.79 CYP2A6 (0.57) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL4772991 0.79 CHRNB2 (0.47) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL3603299 0.79 CYP2A6 (0.68) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL3613286 0.78 CYP2A6 (1.00) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL23781610 0.77 CYP2A6 (0.61) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL29712676 0.76 CHRNB2 (0.66) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL23781611 0.76 HCAR2 (0.43) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8609708-B2 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2013-12-17 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
WO-2005066162-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2005-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer CYP2A13, CYP2A6, CYP2B6 CHRNB2 22/4885CHRNA4 15/4885CYP2A6 2/4885
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER CYP2A13, CYP2A6, CYP2B6 CHRNB2 22/4885CHRNA4 15/4885CYP2A6 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.