SCHEMBL3610698

SCHEMBL3610698

NCc1ccc(-c2cccnc2)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 20/20 1.00
CYP2C19 P33261 16/20 1.00
CYP2E1 P05181 14/20 1.00
CYP2B6 P20813 14/20 1.00
CYP2D6 P10635 13/20 1.00
CYP2C9 P11712 13/20 1.00
CYP3A4 P08684 12/20 1.00
CYP1A2 P05177 8/20 0.73
CYP2C8 P10632 5/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23789552 0.86 CYP2A6 (0.97) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
Hydrochloric Acid SCHEMBL23781581 0.85 CYP2A6 (1.00) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL10162003 0.82 CYP2A6 (0.70) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL13035339 0.82 CYP2A6 (0.70) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL3611935 0.82 CYP2A6 (1.00) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL3615338 0.81 CYP2A6 (1.00) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL31061518 0.81 CYP2A6 (1.00) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL29854440 0.80 CYP2A6 (0.73) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL2690207 0.79 CYP2E1 (1.00) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6
SCHEMBL6513272 0.78 CYP2A6 (0.67) CYP2A6CYP2C19CYP2E1CYP2B6CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-8609708-B2 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2013-12-17 US disclosed
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US disclosed
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2010-11-25 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188527-A1 Synthetic Compounds and Derivatives as Modulators of Smoking or Nicotine Ingestion and Lung Cancer CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP2C19 41/4885CYP2E1 46/4885
US-20100298345-A1 SYNTHETIC COMPOUNDS AND DERIVATIVES AS MODULATORS OF SMOKING OR NICOTINE INGESTION AND LUNG CANCER CYP2A13, CYP2A6, CYP2B6 CYP2A6 2/4885CYP2C19 41/4885CYP2E1 46/4885
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION SLC6A3, NNT, SLC6A2 CYP2A6 1009/4885CYP2C19 3571/4885CYP2E1 1282/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.