SCHEMBL3610798

SCHEMBL3610798

Cc1cccc2cc(C(=O)N[C@H]3CCCNC3)[nH]c12

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.67
NSD2 O96028 3/20 0.62
SETD2 Q9BYW2 2/20 0.62
CHRNA1 P02708 1/20 0.51
CHRNB2 P17787 1/20 0.51
CHRNB4 P30926 1/20 0.51
CHRNA4 P43681 1/20 0.51
HRH4 Q9H3N8 5/20 0.50
PARP1 P09874 1/20 0.47
MAPK1 P28482 1/20 0.46
OPRK1 P41145 1/20 0.46
SYK P43405 1/20 0.46
PLA2G7 Q13093 1/20 0.45
GHSR Q92847 2/20 0.45
CYP1A2 P05177 1/20 0.45
PBK Q96KB5 3/20 0.45
CDK2AP1 O14519 1/20 0.45
CHEK1 O14757 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3610802 1.00 SMYD3 (0.67) SMYD3NSD2SETD2CHRNA1CHRNB2
SCHEMBL3606357 0.93 SMYD3 (0.69) SMYD3NSD2SETD2HRH4PARP1
SCHEMBL3606352 0.93 SMYD3 (0.69) SMYD3NSD2SETD2HRH4PARP1
SCHEMBL3607953 0.93 SMYD3 (0.69) SMYD3NSD2SETD2HRH4PARP1
SCHEMBL21739331 0.87 SMYD3 (0.78) SMYD3NSD2SETD2HRH4PLA2G7
SCHEMBL17209755 0.87 SMYD3 (0.78) SMYD3NSD2SETD2HRH4PLA2G7
SCHEMBL17209750 0.87 SMYD3 (0.78) SMYD3NSD2SETD2HRH4PLA2G7
SCHEMBL3614361 0.86 CDK2 (0.53) SMYD3NSD2SETD2CHRNA1CHRNB2
SCHEMBL3615229 0.86 CDK2 (0.53) SMYD3NSD2SETD2CHRNA1CHRNB2
Trifluoroacetic Acid SCHEMBL3613494 0.86 SMYD3 (0.61) SMYD3NSD2SETD2HRH4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100035862-A1 NOVEL AZA-CYCLIC INDOLE-2-CARBOXAMIDES AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-02-11 US claimed
WO-2009158375-A1 AZA-CYLIC INDOLE- 2 -CARBOXAMIDES AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2009-12-30 WO claimed
US-20100035862-A1 NOVEL AZA-CYCLIC INDOLE-2-CARBOXAMIDES AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-02-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100035862-A1 NOVEL AZA-CYCLIC INDOLE-2-CARBOXAMIDES AND METHODS OF USE THEREOF IDO2, IDO1, INMT SMYD3 811/4885NSD2 146/4885SETD2 2175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.