SCHEMBL361247

SCHEMBL361247

c1cnc(-n2cccn2)c(-c2cn[nH]c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 2/20 0.41
AKT1 P31749 1/20 0.41
FYN P06241 1/20 0.39
AURKA O14965 1/20 0.38
AURKB Q96GD4 1/20 0.38
INCENP Q9NQS7 1/20 0.38
TPX2 Q9ULW0 1/20 0.38
KDM4A O75164 1/20 0.37
KDM4B O94953 1/20 0.37
KDM5C P41229 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
ACVR1B P36896 1/20 0.37
TGFBR1 P36897 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
GRM4 Q14833 1/20 0.35
FEN1 P39748 1/20 0.35
KCNA5 P22460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL320140 0.77 ADORA2A (0.48) KDM4AKDM4BKDM5CKDM5BACVR1B
SCHEMBL361246 0.77 MAPK1 (0.39) AKT2AKT1AURKAAURKBACVR1B
SCHEMBL20534083 0.73 AKT2 (0.50) AKT2AKT1ROCK2MAPK1
SCHEMBL27887721 0.71 ADORA2A (0.43)
SCHEMBL19028096 0.70 AKT1 (0.46) AKT2AKT1FYNAURKAAURKB
SCHEMBL30608796 0.70 AKT1 (0.46) AKT2AKT1FYNAURKAAURKB
SCHEMBL510032 0.70 LRRK2 (0.51) AKT2AKT1FYNAURKAAURKB
Hydrochloric Acid SCHEMBL21806028 0.69 LRRK2 (0.50) AKT2AKT1FYNAURKAAURKB
SCHEMBL21359446 0.69 KDM4E (0.46) AKT2AKT1FYNAURKAAURKB
SCHEMBL2551850 0.69 ADORA2A (0.56) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097594-B2 Macrolides and ketolides having antimicrobial activity WOCKHARDT LTD. (IN) 2012-01-17 US disclosed