SCHEMBL361246

SCHEMBL361246

c1cnc(-c2cn[nH]c2)c(-n2cccn2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.39
NPC1 O15118 1/20 0.39
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
PIM1 P11309 2/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GRM4 Q14833 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
G6PD P11413 1/20 0.36
KMT2A Q03164 1/20 0.36
TDO2 P48775 1/20 0.35
ACVR1B P36896 1/20 0.34
TGFBR1 P36897 1/20 0.34
MPO P05164 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361247 0.77 AKT2 (0.41) MAPK1AKT1AKT2PIM1GRM4
SCHEMBL20534083 0.73 AKT2 (0.50) MAPK1AKT1AKT2KDM4EALDH1A1
SCHEMBL14763854 0.71 NPC1 (0.47) MAPK1NPC1KDM4EALDH1A1MEN1
SCHEMBL30557225 0.70 ALDH1A1 (0.51) MAPK1AKT1AKT2PIM1KDM4E
SCHEMBL29590331 0.70 AKT2 (0.46) MAPK1AKT1AKT2PIM1GRM4
SCHEMBL23291933 0.70 ALDH1A1 (0.51) MAPK1AKT1AKT2PIM1KDM4E
SCHEMBL15308510 0.70 CYP2A6 (0.56) MAPK1AKT1AKT2PIM1KDM4E
SCHEMBL27090965 0.70 AKT2 (0.46) MAPK1AKT1AKT2PIM1GRM4
Hydrochloric Acid SCHEMBL30557160 0.69 ALDH1A1 (0.50) MAPK1AKT1AKT2PIM1KDM4E
Hydrochloric Acid SCHEMBL32685351 0.69 ALDH1A1 (0.50) MAPK1AKT1AKT2PIM1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097594-B2 Macrolides and ketolides having antimicrobial activity WOCKHARDT LTD. (IN) 2012-01-17 US disclosed