Gw7647

Gw7647

SCHEMBL361372

CC(C)(Sc1ccc(CCN(CCCCC2CCCCC2)C(=O)NC2CCCCC2)cc1)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 15/20 1.00
PPARG P37231 13/20 1.00
PPARD Q03181 6/20 1.00
GMNN O75496 1/20 1.00
USP2 O75604 1/20 1.00
USP1 O94782 1/20 1.00
ALDH1A1 P00352 1/20 1.00
LMNA P02545 1/20 1.00
TP53 P04637 1/20 1.00
CYP1A2 P05177 1/20 1.00
POLB P06746 1/20 1.00
CYP3A4 P08684 1/20 1.00
CYP2D6 P10635 1/20 1.00
MAPT P10636 1/20 1.00
CYP2C9 P11712 1/20 1.00
ALOX15 P16050 1/20 1.00
NFKB1 P19838 1/20 1.00
MAPK1 P28482 1/20 1.00
CYP2C19 P33261 1/20 1.00
BRCA1 P38398 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22100299 0.99 PPARA (0.98) PPARAPPARGPPARDGMNNUSP2
SCHEMBL6552622 0.89 PPARA (0.80) PPARAPPARGPPARDGMNNUSP2
SCHEMBL4265257 0.87 PPARA (1.00) PPARAPPARGPPARDGMNNUSP2
SCHEMBL16147204 0.83 PPARA (1.00) PPARAPPARGPPARDGMNNUSP2
SCHEMBL6552333 0.83 PPARA (0.73) PPARAPPARGPPARDGMNNUSP2
SCHEMBL16147851 0.82 PPARA (1.00) PPARAPPARGPPARDGMNNUSP2
SCHEMBL16147225 0.81 PPARA (1.00) PPARAPPARGPPARDGMNNUSP2
SCHEMBL12274271 0.80 PPARA (0.67) PPARAPPARGPPARDGMNNUSP2
SCHEMBL21123888 0.80 PPARA (0.67) PPARAPPARGPPARDGMNNUSP2
SCHEMBL3675079 0.79 PPARA (0.65) PPARAPPARGPPARDGMNNUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 815 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4725479-A1 PPAR AGONISTS FOR TREATMENT OF DISEASES ASSOCIATED WITH AATD Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2026-04-15 EP claimed
US-20250297321-A1 METHOD FOR DETECTING METABOLIC REPROGRAMING OF CANCER TOWARDS FATTY ACIDS METABOLISM INST NAT SANTE RECH MED (FR) 2025-09-25 US claimed
EP-4583859-A2 COMPOSITIONS FOR PREVENTING TRANSITION FROM ACUTE TO CHRONIC PAIN The Regents of University of California (US) 2025-07-16 EP claimed
EP-4558622-A1 METHODS AND COMPOSITIONS FOR GENERATING HUMAN MIDBRAIN DOPAMINERGIC NEURONS FROM NEURAL PROGENITOR CELLS Trailhead Biosystems Inc. (US) 2025-05-28 EP claimed
CN-120051560-A Methods and compositions for generating human midbrain dopaminergic neurons from neural progenitor cells 特雷尔赫德生物系统股份有限公司 2025-05-27 CN claimed
CN-120004949-A Mitochondria targeting compound, preparation method and application thereof, and pharmaceutical composition 中国医学科学院医药生物技术研究所 2025-05-16 CN claimed
CN-119235836-A Application of GW7647 in preparation of medicine for inhibiting cell lipid peroxidation caused by African swine fever virus protein 华中农业大学 2025-01-03 CN claimed
US-20240398789-A1 PHARMACEUTICAL COMPOSITION FOR ENHANCING ANTI-TUMOR EFFECT OF EZH2 INHIBITOR AND USE THEREOF PEKING UNIVERSITY THIRD HOSPITAL (CN) 2024-12-05 US claimed
EP-4469602-A1 METHOD FOR DETECTING METABOLIC REPROGRAMING OF CANCER TOWARDS FATTY ACIDS METABOLISM Université Paris Cité (FR) 2024-12-04 EP claimed
US-20240285540-A1 FUNCTIONAL THERAPEUTIC INDEX IN THE TREATMENT OF PERIPHERAL IMMUNE DYSFUNCTION MASCARENHAS DESMOND (US) 2024-08-29 US claimed
EP-1569640-A4 COMBINATIONS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR-ALPHA AGONISTS AND CYCLOOXYGENASE-2 SELECTIVE INHIBITORS AND THERAPEUTIC USES THEREFOR PHARMACIA CORP (US) 2006-06-21 EP claimed
EP-1569640-A2 COMBINATIONS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR-ALPHA AGONISTS AND CYCLOOXYGENASE-2 SELECTIVE INHIBITORS AND THERAPEUTIC USES THEREFOR Pharmacia Corporation (US) 2005-09-07 EP claimed
US-20050054730-A1 Compounds, compositions and treatment of oleoylethanolamide-like modulators of PPARalpha THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2005-03-10 US claimed
WO-2005002524-A2 COMPOUNDS, COMPOSITIONS AND THERAPEUTIC USES OF OLEOYLETHANOLAMIDE-LIKE COMPOUNDS AND MODULATORS OF PPARα THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2005-01-13 WO claimed
EP-1149063-B1 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS SMITHKLINE BEECHAM CORP (US) 2004-12-15 EP claimed
US-20030212138-A1 Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2 selective inhibitors and therapeutic uses therefor PHARMACIA CORPORATION (US) 2003-11-13 US claimed
WO-2003059294-A2 COMBINATIONS OF PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR-ALPHA AGONISTS AND CYCLOOXYGENASE-2 SELECTIVE INHIBITORS AND THERAPEUTIC USES THEREFOR PHARMACIA CORPORATION (US) 2003-07-24 WO claimed
EP-1149063-A2 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS GLAXO GROUP LIMITED (GB) 2001-10-31 EP claimed
US-6306854-B1 ARYLTHIOALKYLACIDS AND ALKYL UREAS GLAXOSMITHKLINE 2001-10-23 US claimed
WO-2000023407-A2 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS GLAXO GROUP LIMITED (GB) 2000-04-27 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030212138-A1 Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2 selective inhibitors and therapeutic uses therefor PPARG, PPARA, PPARD PPARA 2/4885PPARG 1/4885PPARD 3/4885
US-20050054730-A1 Compounds, compositions and treatment of oleoylethanolamide-like modulators of PPARalpha PPARA, CNR2, CNR1 PPARA 1/4885PPARG 11/4885PPARD 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.